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Belladonna Alkaloids Ergotamine Phenobarbital Brand Names
Bel Phen Ergot | Bel Tabs | Bellamine | Bellamine S | Bellaspas | Bellergal-S | Eperbel-S | Spastrin
What is Belladonna Alkaloids Ergotamine Phenobarbital
NOTE: These products are discontinued in the U.S.
Belladonna Alkaloids Ergotamine Phenobarbital is used as a prophylaxis for migraine and vascular headaches.
Historically, this autonomic drug combination was used in the non-specific treatment of various gastrointestinal, genitourinary, and cardiovascular disorders but has been replaced with more medically specific and effective therapies for such conditions.
Belladonna alkaloids; ergotamine; phenobarbital products have been employed since pre-1938 for the management of disorders characterized by nervous tension and exaggerated autonomic response.
It has also been used clinically for many years to relieve climacteric symptoms in females with contraindications to traditional hormone replacement therapy (HRT) or those that choose not to take HRT.
Indications
- menopause
- migraine prophylaxis
For migraine prophylaxis or vascular headache prophylaxis
Side Effects
- abdominal pain
- agitation
- agranulocytosis
- anemia
- angina
- angioedema
- anhidrosis
- anxiety
- asthenia
- ataxia
- blurred vision
- bone pain
- bradycardia
- bullous rash
- cardiac valvulopathy
- chest pain (unspecified)
- colitis
- coma
- confusion
- constipation
- coronary vasospasm
- cycloplegia
- delirium
- depression
- dizziness
- drowsiness
- dyspepsia
- dysphagia
- ecchymosis
- edema
- elevated hepatic enzymes
- emotional lability
- exfoliative dermatitis
- fatigue
- fetal death
- fever
- flushing
- hallucinations
- headache
- hepatitis
- hypoprothrombinemia
- hypotension
- hypothermia
- ileus
- impaired cognition
- impotence (erectile dysfunction)
- insomnia
- interstitial nephritis
- irritability
- jaundice
- lethargy
- libido decrease
- lupus-like symptoms
- maculopapular rash
- megaloblastic anemia
- miosis
- muscle cramps
- myalgia
- mydriasis
- myocardial infarction
- nausea
- neonatal abstinence syndrome
- neutropenia
- nightmares
- nystagmus
- ocular hypertension
- osteomalacia
- osteopenia
- palpitations
- pancreatitis
- paresthesias
- peripheral vasoconstriction
- photophobia
- photosensitivity
- physiological dependence
- porphyria
- pruritus
- psychological dependence
- ptosis
- pulmonary fibrosis
- purpura
- pyrosis (heartburn)
- renal tubular necrosis
- respiratory depression
- retroperitoneal fibrosis
- seizures
- serum sickness
- sinus tachycardia
- spontaneous fetal abortion
- Stevens-Johnson syndrome
- teratogenesis
- thrombocytopenia
- thrombosis
- tissue necrosis
- tolerance
- toxic epidermal necrolysis
- urinary retention
- urticaria
- uterine contractions
- vertigo
- vomiting
- weakness
- weight loss
- withdrawal
- xerostomia
Monitoring Parameters
- CBC
- LFTs
- serum creatinine/BUN
Contraindications
- abrupt discontinuation
- achalasia
- acute myocardial infarction
- ambient temperature increase
- angina
- anticoagulant therapy
- arteriosclerosis
- asthma
- autonomic neuropathy
- barbiturate hypersensitivity
- basilar/hemiplegic migraine
- biliary tract disease
- bladder obstruction
- bleeding
- breast-feeding
- carbamazepine hypersensitivity
- cardiac arrhythmias
- cardiac disease
- children
- cholestasis
- chronic obstructive pulmonary disease (COPD)
- closed-angle glaucoma
- colostomy
- contact lenses
- coronary artery disease
- dehydration
- dental disease
- depression
- diabetes mellitus
- diarrhea
- driving or operating machinery
- ergot alkaloid hypersensitivity
- esophagitis
- ethanol ingestion
- fever
- gastroesophageal reflux disease (GERD)
- geriatric
- GI disease
- GI obstruction
- glaucoma
- heart failure
- hepatic disease
- hiatal hernia
- hydantoin hypersensitivity
- hypercholesterolemia
- hypertension
- hyperthyroidism
- ileostomy
- ileus
- infants
- labor
- mental status changes
- mitral stenosis
- myasthenia gravis
- obesity
- obstetric delivery
- peptic ulcer disease
- peripheral vascular disease
- porphyria
- pregnancy
- prostatic hypertrophy
- pseudomembranous colitis
- pulmonary disease
- pulmonary fibrosis
- pyloric stenosis
- Raynaud’s phenomenon
- renal disease
- renal failure
- renal impairment
- respiratory depression
- respiratory infection
- respiratory insufficiency
- retroperitoneal fibrosis
- sepsis
- shock
- strenuous exercise
- stroke
- substance abuse
- suicidal ideation
- surgery
- synechia
- tachycardia
- thromboangiitis obliterans (Buerger’s disease)
- thrombophlebitis
- thyrotoxicosis
- tobacco smoking
- toxic megacolon
- ulcerative colitis
- urinary retention
- urinary tract obstruction
- valvular heart disease
Interactions
- Abacavir; Dolutegravir; Lamivudine
- Abemaciclib
- Abiraterone
- Acalabrutinib
- Acebutolol
- Acetaminophen
- Acetaminophen; Aspirin, ASA; Caffeine
- Acetaminophen; Butalbital
- Acetaminophen; Butalbital; Caffeine
- Acetaminophen; Butalbital; Caffeine; Codeine
- Acetaminophen; Caffeine
- Acetaminophen; Caffeine; Dihydrocodeine
- Acetaminophen; Caffeine; Magnesium Salicylate; Phenyltoloxamine
- Acetaminophen; Caffeine; Phenyltoloxamine; Salicylamide
- Acetaminophen; Chlorpheniramine; Dextromethorphan; Phenylephrine
- Acetaminophen; Chlorpheniramine; Dextromethorphan; Pseudoephedrine
- Acetaminophen; Chlorpheniramine; Phenylephrine; Phenyltoloxamine
- Acetaminophen; Codeine
- Acetaminophen; Dextromethorphan
- Acetaminophen; Dextromethorphan; Doxylamine
- Acetaminophen; Dextromethorphan; Guaifenesin; Phenylephrine
- Acetaminophen; Dextromethorphan; Phenylephrine
- Acetaminophen; Dextromethorphan; Pseudoephedrine
- Acetaminophen; Dichloralphenazone; Isometheptene
- Acetaminophen; Diphenhydramine
- Acetaminophen; Guaifenesin; Phenylephrine
- Acetaminophen; Hydrocodone
- Acetaminophen; Oxycodone
- Acetaminophen; Pentazocine
- Acetaminophen; Propoxyphene
- Acetaminophen; Pseudoephedrine
- Acetaminophen; Tramadol
- Acetazolamide
- Aclidinium
- Aclidinium; Formoterol
- Acrivastine; Pseudoephedrine
- Afatinib
- Albendazole
- Albuterol; Ipratropium
- Aldesleukin, IL-2
- Alfentanil
- Aliskiren; Amlodipine
- Aliskiren; Amlodipine; Hydrochlorothiazide, HCTZ
- Aliskiren; Hydrochlorothiazide, HCTZ
- Almotriptan
- Alogliptin; Pioglitazone
- Alosetron
- Alpelisib
- Alprazolam
- Altretamine
- Aluminum Hydroxide
- Aluminum Hydroxide; Magnesium Carbonate
- Aluminum Hydroxide; Magnesium Hydroxide
- Aluminum Hydroxide; Magnesium Hydroxide; Simethicone
- Aluminum Hydroxide; Magnesium Trisilicate
- Amiloride; Hydrochlorothiazide, HCTZ
- Aminosalicylate sodium, Aminosalicylic acid
- Amiodarone
- Amitriptyline; Chlordiazepoxide
- Amlodipine
- Amlodipine; Atorvastatin
- Amlodipine; Benazepril
- Amlodipine; Celecoxib
- Amlodipine; Hydrochlorothiazide, HCTZ; Olmesartan
- Amlodipine; Hydrochlorothiazide, HCTZ; Valsartan
- Amlodipine; Olmesartan
- Amlodipine; Telmisartan
- Amlodipine; Valsartan
- Amoxapine
- Amoxicillin; Clarithromycin; Lansoprazole
- Amoxicillin; Clarithromycin; Omeprazole
- Amphetamine
- Amphetamine; Dextroamphetamine
- Amphetamine; Dextroamphetamine Salts
- Amprenavir
- Anagrelide
- Antacids
- Apixaban
- Apomorphine
- Apraclonidine
- Apremilast
- Aprepitant, Fosaprepitant
- Aripiprazole
- Armodafinil
- Artemether; Lumefantrine
- Articaine; Epinephrine
- Asenapine
- Aspirin, ASA
- Aspirin, ASA; Butalbital; Caffeine
- Aspirin, ASA; Butalbital; Caffeine; Codeine
- Aspirin, ASA; Caffeine; Dihydrocodeine
- Aspirin, ASA; Caffeine; Orphenadrine
- Aspirin, ASA; Carisoprodol
- Aspirin, ASA; Carisoprodol; Codeine
- Aspirin, ASA; Citric Acid; Sodium Bicarbonate
- Aspirin, ASA; Dipyridamole
- Aspirin, ASA; Omeprazole
- Aspirin, ASA; Oxycodone
- Aspirin, ASA; Pravastatin
- Atazanavir
- Atazanavir; Cobicistat
- Atenolol
- Atenolol; Chlorthalidone
- Atorvastatin
- Atorvastatin; Ezetimibe
- Atropine; Benzoic Acid; Hyoscyamine; Methenamine; Methylene Blue; Phenyl Salicylate
- Atropine; Difenoxin
- Atropine; Diphenoxylate
- Atropine; Hyoscyamine; Phenobarbital; Scopolamine
- Avanafil
- Avapritinib
- Avatrombopag
- Axitinib
- Azelastine
- Azelastine; Fluticasone
- Azilsartan; Chlorthalidone
- Azithromycin
- Bedaquiline
- Belladonna; Opium
- Benazepril; Hydrochlorothiazide, HCTZ
- Bendamustine
- Bendroflumethiazide; Nadolol
- Benzhydrocodone; Acetaminophen
- Benzoic Acid; Hyoscyamine; Methenamine; Methylene Blue; Phenyl Salicylate
- Benzphetamine
- Benztropine
- Beta-blockers
- Betaxolol
- Betrixaban
- Bicalutamide
- Bictegravir; Emtricitabine; Tenofovir Alafenamide
- Biotin
- Bismuth Subcitrate Potassium; Metronidazole; Tetracycline
- Bismuth Subsalicylate
- Bismuth Subsalicylate; Metronidazole; Tetracycline
- Bisoprolol
- Bisoprolol; Hydrochlorothiazide, HCTZ
- Boceprevir
- Bortezomib
- Bosentan
- Bosutinib
- Botulinum Toxins
- Brentuximab vedotin
- Brexpiprazole
- Brigatinib
- Brimonidine
- Brimonidine; Brinzolamide
- Brimonidine; Timolol
- Brivaracetam
- Bromocriptine
- Brompheniramine
- Brompheniramine; Carbetapentane; Phenylephrine
- Brompheniramine; Dextromethorphan; Guaifenesin
- Brompheniramine; Guaifenesin; Hydrocodone
- Brompheniramine; Hydrocodone; Pseudoephedrine
- Brompheniramine; Pseudoephedrine
- Budesonide
- Budesonide; Formoterol
- Bupivacaine
- Bupivacaine Liposomal
- Bupivacaine; Lidocaine
- Buprenorphine
- Buprenorphine; Naloxone
- Bupropion
- Bupropion; Naltrexone
- Buspirone
- Butorphanol
- Cabergoline
- Cabozantinib
- Caffeine
- Caffeine; Ergotamine
- Calcifediol
- Calcitriol
- Calcium Carbonate
- Calcium Carbonate; Magnesium Hydroxide
- Calcium Carbonate; Risedronate
- Calcium Carbonate; Simethicone
- Canagliflozin
- Canagliflozin; Metformin
- Canakinumab
- Candesartan; Hydrochlorothiazide, HCTZ
- Cannabidiol
- Capmatinib
- Captopril; Hydrochlorothiazide, HCTZ
- Carbamazepine
- Carbetapentane; Chlorpheniramine
- Carbetapentane; Chlorpheniramine; Phenylephrine
- Carbetapentane; Diphenhydramine; Phenylephrine
- Carbetapentane; Guaifenesin
- Carbetapentane; Guaifenesin; Phenylephrine
- Carbetapentane; Phenylephrine
- Carbetapentane; Phenylephrine; Pyrilamine
- Carbetapentane; Pseudoephedrine
- Carbetapentane; Pyrilamine
- Carbidopa; Levodopa
- Carbidopa; Levodopa; Entacapone
- Carbinoxamine
- Carbinoxamine; Dextromethorphan; Pseudoephedrine
- Carbinoxamine; Hydrocodone; Phenylephrine
- Carbinoxamine; Hydrocodone; Pseudoephedrine
- Carbinoxamine; Phenylephrine
- Carbinoxamine; Pseudoephedrine
- Cardiac glycosides
- Cariprazine
- Carmustine, BCNU
- Carteolol
- Carvedilol
- Cenobamate
- Ceritinib
- Cetirizine
- Cetirizine; Pseudoephedrine
- Cevimeline
- Chlophedianol; Dexbrompheniramine
- Chlophedianol; Dexchlorpheniramine; Pseudoephedrine
- Chlorambucil
- Chloramphenicol
- Chlorcyclizine
- Chlordiazepoxide
- Chlordiazepoxide; Clidinium
- Chloroprocaine
- Chloroquine
- Chlorothiazide
- Chlorpheniramine
- Chlorpheniramine; Codeine
- Chlorpheniramine; Dextromethorphan
- Chlorpheniramine; Dextromethorphan; Phenylephrine
- Chlorpheniramine; Dihydrocodeine; Phenylephrine
- Chlorpheniramine; Dihydrocodeine; Pseudoephedrine
- Chlorpheniramine; Guaifenesin; Hydrocodone; Pseudoephedrine
- Chlorpheniramine; Hydrocodone
- Chlorpheniramine; Hydrocodone; Phenylephrine
- Chlorpheniramine; Hydrocodone; Pseudoephedrine
- Chlorpheniramine; Phenylephrine
- Chlorpheniramine; Pseudoephedrine
- Chlorpromazine
- Chlorthalidone
- Chlorthalidone; Clonidine
- Choline Salicylate; Magnesium Salicylate
- Cholinergic agonists
- Cimetidine
- Cinacalcet
- Citalopram
- Clarithromycin
- Clemastine
- Clindamycin
- Clobazam
- Clofazimine
- Clonazepam
- Clopidogrel
- Clorazepate
- Clozapine
- Cobicistat
- Cobimetinib
- Cocaine
- Codeine
- Codeine; Guaifenesin
- Codeine; Phenylephrine; Promethazine
- Codeine; Promethazine
- Colesevelam
- COMT inhibitors
- Conivaptan
- Conjugated Estrogens
- Conjugated Estrogens; Bazedoxifene
- Conjugated Estrogens; Medroxyprogesterone
- Copanlisib
- Crizotinib
- Crofelemer
- Cyclizine
- Cyclobenzaprine
- Cyclophosphamide
- Cyclosporine
- Cyproheptadine
- Dabigatran
- Dabrafenib
- Daclatasvir
- Danazol
- Dapagliflozin
- Dapagliflozin; Metformin
- Dapagliflozin; Saxagliptin
- Dapsone
- Darifenacin
- Darolutamide
- Darunavir
- Darunavir; Cobicistat
- Darunavir; Cobicistat; Emtricitabine; Tenofovir alafenamide
- Dasabuvir; Ombitasvir; Paritaprevir; Ritonavir
- Dasatinib
- Deferasirox
- Deflazacort
- Delavirdine
- Desloratadine; Pseudoephedrine
- Desvenlafaxine
- Deutetrabenazine
- Dexamethasone
- Dexchlorpheniramine
- Dexchlorpheniramine; Dextromethorphan; Pseudoephedrine
- Dexlansoprazole
- Dexmedetomidine
- Dextroamphetamine
- Dextromethorphan; Diphenhydramine; Phenylephrine
- Dextromethorphan; Guaifenesin; Pseudoephedrine
- Dextromethorphan; Promethazine
- Dextromethorphan; Quinidine
- Diazepam
- Diazoxide
- Diclofenac
- Diclofenac; Misoprostol
- Dicyclomine
- Dienogest; Estradiol valerate
- Diethylstilbestrol, DES
- Dihydrocodeine; Guaifenesin; Pseudoephedrine
- Diltiazem
- Dimenhydrinate
- Diphenhydramine
- Diphenhydramine; Hydrocodone; Phenylephrine
- Diphenhydramine; Ibuprofen
- Diphenhydramine; Naproxen
- Diphenhydramine; Phenylephrine
- Dirithromycin
- Disopyramide
- Dobutamine
- Docetaxel
- Dolutegravir
- Dolutegravir; Lamivudine
- Dolutegravir; Rilpivirine
- Donepezil
- Donepezil; Memantine
- Doravirine
- Doravirine; Lamivudine; Tenofovir disoproxil fumarate
- Dorzolamide; Timolol
- Doxercalciferol
- Doxorubicin
- Doxycycline
- Doxylamine
- Doxylamine; Pyridoxine
- Dronabinol
- Dronedarone
- Droperidol
- Drospirenone; Estradiol
- Drospirenone; Ethinyl Estradiol
- Drospirenone; Ethinyl Estradiol; Levomefolate
- Duloxetine
- Duvelisib
- Edoxaban
- Efavirenz
- Efavirenz; Emtricitabine; Tenofovir
- Efavirenz; Lamivudine; Tenofovir Disoproxil Fumarate
- Elagolix
- Elagolix; Estradiol; Norethindrone acetate
- Elbasvir; Grazoprevir
- Eletriptan
- Elexacaftor; tezacaftor; ivacaftor
- Eliglustat
- Eltrombopag
- Eluxadoline
- Elvitegravir
- Elvitegravir; Cobicistat; Emtricitabine; Tenofovir Alafenamide
- Elvitegravir; Cobicistat; Emtricitabine; Tenofovir Disoproxil Fumarate
- Emapalumab
- Empagliflozin; Linagliptin
- Empagliflozin; Linagliptin; Metformin
- Emtricitabine; Rilpivirine; Tenofovir alafenamide
- Emtricitabine; Rilpivirine; Tenofovir disoproxil fumarate
- Emtricitabine; Tenofovir alafenamide
- Enalapril; Felodipine
- Enalapril; Hydrochlorothiazide, HCTZ
- Encorafenib
- Entacapone
- Entrectinib
- Enzalutamide
- Epinephrine
- Eprosartan; Hydrochlorothiazide, HCTZ
- Eravacycline
- Erdafitinib
- Erlotinib
- Erythromycin
- Erythromycin; Sulfisoxazole
- Escitalopram
- Esketamine
- Eslicarbazepine
- Esmolol
- Esomeprazole
- Esomeprazole; Naproxen
- Estazolam
- Esterified Estrogens
- Esterified Estrogens; Methyltestosterone
- Estradiol
- Estradiol Cypionate; Medroxyprogesterone
- Estradiol; Levonorgestrel
- Estradiol; Norethindrone
- Estradiol; Norgestimate
- Estradiol; Progesterone
- Estrogens
- Estropipate
- Eszopiclone
- Ethanol
- Ethinyl Estradiol
- Ethinyl Estradiol; Desogestrel
- Ethinyl Estradiol; Ethynodiol Diacetate
- Ethinyl Estradiol; Etonogestrel
- Ethinyl Estradiol; Levonorgestrel
- Ethinyl Estradiol; Levonorgestrel; Ferrous bisglycinate
- Ethinyl Estradiol; Levonorgestrel; Folic Acid; Levomefolate
- Ethinyl Estradiol; Norelgestromin
- Ethinyl Estradiol; Norethindrone
- Ethinyl Estradiol; Norethindrone Acetate
- Ethinyl Estradiol; Norethindrone Acetate; Ferrous fumarate
- Ethinyl Estradiol; Norethindrone; Ferrous fumarate
- Ethinyl Estradiol; Norgestimate
- Ethinyl Estradiol; Norgestrel
- Ethosuximide
- Etravirine
- Everolimus
- Exemestane
- Ezetimibe; Simvastatin
- Ezogabine
- Fedratinib
- Felbamate
- Felodipine
- Fenofibric Acid
- Fenoldopam
- Fenoprofen
- Fentanyl
- Fexofenadine; Pseudoephedrine
- Flibanserin
- Fluconazole
- Fluoxetine
- Fluoxetine; Olanzapine
- Fluphenazine
- Fluticasone
- Fluticasone; Salmeterol
- Fluticasone; Umeclidinium; Vilanterol
- Fluticasone; Vilanterol
- Fluvoxamine
- Folic Acid, Vitamin B9
- food
- Fosamprenavir
- Fosinopril; Hydrochlorothiazide, HCTZ
- Fostamatinib
- Frovatriptan
- Gabapentin
- Galantamine
- Gallium Ga 68 Dotatate
- Gefitinib
- General anesthetics
- Gilteritinib
- Glasdegib
- Glecaprevir; Pibrentasvir
- Glimepiride
- Glimepiride; Pioglitazone
- Glimepiride; Rosiglitazone
- Glucagon
- Glycerol Phenylbutyrate
- Glycopyrronium
- Granisetron
- grapefruit juice
- Green Tea
- Griseofulvin
- Guaifenesin; Hydrocodone
- Guaifenesin; Hydrocodone; Pseudoephedrine
- Guaifenesin; Pseudoephedrine
- Guanfacine
- Haloperidol
- Hemin
- Homatropine; Hydrocodone
- Hydantoins
- Hydralazine
- Hydralazine; Hydrochlorothiazide, HCTZ
- Hydralazine; Isosorbide Dinitrate, ISDN
- Hydrochlorothiazide, HCTZ
- Hydrochlorothiazide, HCTZ; Irbesartan
- Hydrochlorothiazide, HCTZ; Lisinopril
- Hydrochlorothiazide, HCTZ; Losartan
- Hydrochlorothiazide, HCTZ; Methyldopa
- Hydrochlorothiazide, HCTZ; Metoprolol
- Hydrochlorothiazide, HCTZ; Moexipril
- Hydrochlorothiazide, HCTZ; Olmesartan
- Hydrochlorothiazide, HCTZ; Propranolol
- Hydrochlorothiazide, HCTZ; Quinapril
- Hydrochlorothiazide, HCTZ; Spironolactone
- Hydrochlorothiazide, HCTZ; Telmisartan
- Hydrochlorothiazide, HCTZ; Triamterene
- Hydrochlorothiazide, HCTZ; Valsartan
- Hydrocodone
- Hydrocodone; Ibuprofen
- Hydrocodone; Phenylephrine
- Hydrocodone; Potassium Guaiacolsulfonate
- Hydrocodone; Potassium Guaiacolsulfonate; Pseudoephedrine
- Hydrocodone; Pseudoephedrine
- Hydromorphone
- Hydroxychloroquine
- Hydroxyzine
- Hyoscyamine; Methenamine; Methylene Blue; Phenyl Salicylate; Sodium Biphosphate
- Ibrutinib
- Ibuprofen; Oxycodone
- Ibuprofen; Pseudoephedrine
- Idelalisib
- Ifosfamide
- Iloperidone
- Imatinib
- Indinavir
- Indocyanine Green
- Ipratropium
- Irinotecan
- Irinotecan Liposomal
- Isavuconazonium
- Isocarboxazid
- Isoniazid, INH; Pyrazinamide, PZA; Rifampin
- Isoniazid, INH; Rifampin
- Isoproterenol
- Isradipine
- Istradefylline
- Itraconazole
- Ivabradine
- Ivacaftor
- Ivosidenib
- Ixabepilone
- Ixazomib
- Ketoconazole
- Labetalol
- Lamotrigine
- Lanreotide
- Lansoprazole
- Lansoprazole; Naproxen
- Lapatinib
- Larotrectinib
- Lasmiditan
- Ledipasvir; Sofosbuvir
- Lefamulin
- Lemborexant
- Lesinurad
- Lesinurad; Allopurinol
- Letermovir
- Leucovorin
- Levobetaxolol
- Levobunolol
- Levobupivacaine
- Levocetirizine
- Levodopa
- Levoleucovorin
- Levomefolate
- Levomilnacipran
- Levorphanol
- Lidocaine
- Lidocaine; Prilocaine
- Linaclotide
- Linagliptin
- Linagliptin; Metformin
- Linezolid
- Lisdexamfetamine
- Lithium
- Lofexidine
- Lomustine, CCNU
- Loperamide
- Loperamide; Simethicone
- Lopinavir; Ritonavir
- Loratadine; Pseudoephedrine
- Lorazepam
- Lorcaserin
- Lorlatinib
- Losartan
- Lovastatin
- Lovastatin; Niacin
- Loxapine
- Lubiprostone
- Lumacaftor; Ivacaftor
- Lumacaftor; Ivacaftor
- Lumateperone
- Lurasidone
- Lurbinectedin
- Macimorelin
- Magnesium Hydroxide
- Magnesium Salicylate
- Magnesium Salts
- Mannitol
- Maprotiline
- Maraviroc
- Mebendazole
- Meclizine
- Mefloquine
- Melatonin
- Memantine
- Meperidine
- Meperidine; Promethazine
- Mepivacaine
- Mepivacaine; Levonordefrin
- Meprobamate
- Mestranol; Norethindrone
- Metformin; Pioglitazone
- Metformin; Repaglinide
- Methacholine
- Methadone
- Methamphetamine
- Methazolamide
- Methenamine; Sodium Acid Phosphate; Methylene Blue; Hyoscyamine
- Methocarbamol
- Methscopolamine
- Methsuximide
- Methyclothiazide
- Methylene Blue
- Methylphenidate
- Methylprednisolone
- Metoclopramide
- Metolazone
- Metoprolol
- Metronidazole
- Metyrapone
- Metyrosine
- Mexiletine
- Miconazole
- Midazolam
- Midostaurin
- Mifepristone
- Milnacipran
- Minocycline
- Minoxidil
- Mirtazapine
- Mitotane
- Modafinil
- Molindone
- Monoamine oxidase inhibitors
- Montelukast
- Morphine
- Morphine; Naltrexone
- Nabilone
- Nadolol
- Nalbuphine
- Naldemedine
- Naloxegol
- Nanoparticle Albumin-Bound Paclitaxel
- Naproxen; Pseudoephedrine
- Naproxen; Sumatriptan
- Naratriptan
- Nebivolol
- Nebivolol; Valsartan
- Nefazodone
- Nelfinavir
- Neratinib
- Netupitant, Fosnetupitant; Palonosetron
- Nevirapine
- Niacin; Simvastatin
- Nicardipine
- Nicotine
- Nifedipine
- Nilotinib
- Nimodipine
- Nintedanib
- Nisoldipine
- Nitrates
- Nitrofurantoin
- Nitroprusside
- Norfloxacin
- Olanzapine
- Olaparib
- Ombitasvir; Paritaprevir; Ritonavir
- Omeprazole
- Omeprazole; Amoxicillin; Rifabutin
- Omeprazole; Sodium Bicarbonate
- Ondansetron
- Oritavancin
- Osilodrostat
- Osimertinib
- Ospemifene
- Oxazepam
- Oxcarbazepine
- Oxybutynin
- Oxycodone
- Oxymorphone
- Paclitaxel
- Palbociclib
- Paliperidone
- Panobinostat
- Papaverine
- Paroxetine
- Pazopanib
- Pemoline
- Penbutolol
- Penicillin G Benzathine; Penicillin G Procaine
- Penicillin G Procaine
- Pentazocine
- Pentazocine; Naloxone
- Perampanel
- Perindopril; Amlodipine
- Perphenazine
- Perphenazine; Amitriptyline
- Pexidartinib
- Phenelzine
- Phenothiazines
- Phentermine
- Phentermine; Topiramate
- Phenylephrine; Promethazine
- Pimavanserin
- Pindolol
- Pioglitazone
- Pitolisant
- Polatuzumab Vedotin
- Pomalidomide
- Ponatinib
- Posaconazole
- Potassium
- Pralidoxime
- Pramipexole
- Pramlintide
- Praziquantel
- Prednisolone
- Prednisone
- Pregabalin
- Prilocaine
- Prilocaine; Epinephrine
- Procainamide
- Procaine
- Procarbazine
- Prochlorperazine
- Progestins
- Promethazine
- Propranolol
- Protease inhibitors
- Proton pump inhibitors
- Pseudoephedrine
- Pyridoxine, Vitamin B6
- Quazepam
- Quetiapine
- Quinidine
- Quinine
- Rabeprazole
- Raltegravir
- Ramelteon
- Ranolazine
- Rasagiline
- Red Yeast Rice
- Regorafenib
- Remdesivir
- Remifentanil
- Repaglinide
- Reserpine
- Revefenacin
- Ribociclib
- Ribociclib; Letrozole
- Rifampin
- Rifapentine
- Rilpivirine
- Riluzole
- Rimegepant
- Riociguat
- Ripretinib
- Risperidone
- Ritonavir
- Rivaroxaban
- Rivastigmine
- Rizatriptan
- Roflumilast
- Rolapitant
- Romidepsin
- Ropinirole
- Ropivacaine
- Rotigotine
- Rucaparib
- Rufinamide
- Ruxolitinib
- Safinamide
- Salicylates
- Salsalate
- Sapropterin
- Saquinavir
- Sarilumab
- Scopolamine
- Secretin
- Sedating H1-blockers
- Segesterone Acetate; Ethinyl Estradiol
- Selegiline
- Selpercatinib
- Selumetinib
- Serotonin norepinephrine reuptake inhibitors
- Serotonin-Receptor Agonists
- Sertraline
- Sibutramine
- Sildenafil
- Siltuximab
- Simeprevir
- Simvastatin
- Simvastatin; Sitagliptin
- Sincalide
- Siponimod
- Sirolimus
- Skeletal Muscle Relaxants
- Sodium Bicarbonate
- Sodium Oxybate
- Sofosbuvir
- Sofosbuvir; Velpatasvir
- Sofosbuvir; Velpatasvir; Voxilaprevir
- Solifenacin
- Sonidegib
- Sorafenib
- Sotalol
- Spironolactone
- Streptogramins
- Sufentanil
- Sumatriptan
- Sunitinib
- Suvorexant
- Tacrine
- Tacrolimus
- Tadalafil
- Tamoxifen
- Tapentadol
- Tasimelteon
- Tazemetostat
- Tedizolid
- Tegaserod
- Telaprevir
- Telithromycin
- Telotristat Ethyl
- Temazepam
- Temsirolimus
- Teniposide
- Tenofovir Alafenamide
- Tenofovir Alafenamide
- Terbinafine
- Tetrabenazine
- Tetracaine
- Tezacaftor; Ivacaftor
- Thalidomide
- Theophylline, Aminophylline
- Thiazide diuretics
- Thioridazine
- Thiotepa
- Thiothixene
- Thyroid hormones
- Tiagabine
- Ticagrelor
- Timolol
- Tinidazole
- Tiotropium
- Tiotropium; Olodaterol
- Tipranavir
- Tizanidine
- tobacco
- Tocilizumab
- Tofacitinib
- Tolcapone
- Tolterodine
- Tolvaptan
- Topiramate
- Toremifene
- Trabectedin
- Tramadol
- Trandolapril; Verapamil
- Tranylcypromine
- Trazodone
- Tretinoin, ATRA
- Triamcinolone
- Triazolam
- Tricyclic antidepressants
- Trifluoperazine
- Trimethobenzamide
- Trimetrexate
- Triprolidine
- Trospium
- Tucatinib
- Ubrogepant
- Ulipristal
- Umeclidinium
- Umeclidinium; Vilanterol
- Upadacitinib
- Valbenazine
- Valerian, Valeriana officinalis
- Valproic Acid, Divalproex Sodium
- Vandetanib
- Vasopressors
- Vemurafenib
- Venetoclax
- Venlafaxine
- Verapamil
- Vigabatrin
- Vilazodone
- Vincristine
- Vincristine Liposomal
- Vorapaxar
- Voriconazole
- Vortioxetine
- Voxelotor
- Warfarin
- Zafirlukast
- Zaleplon
- Zanubrutinib
- Ziconotide
- Zileuton
- Ziprasidone
- Zolmitriptan
- Zolpidem
- Zonisamide