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Aspirin Butalbital Caffeine Brand Names- Fiorinal | Fortabs
What is Aspirin Butalbital Caffeine
Aspirin butalbital caffeine are used together in an oral preparation to treat tension headaches, migraines, and mild to moderate pain, especially when antianxiety or relaxant effects are needed.
Treatment of multiple recurrent headaches with this combination has not been well studied.
According to published guidelines for the acute management of migraine, the use of butalbital-containing analgesics should be limited and carefully monitored due to concerns of overuse, medication-overuse headache, and withdrawal.
Aspirin is a salicylate analgesic with similar analgesic potency to NSAIDs. Butalbital is a short-to-intermediate acting barbiturate that is used in this combination for its sedative and relaxant effects.
Caffeine is found in many analgesic formulations and may be beneficial in some vascular headaches such as tension and cluster headaches and migraines.
Fiorinal was originally approved by the FDA in May 1976.
Indications
- headache
- migraine
For the treatment of occasional tension headache, occasional migraine† or co-existing migraine† and tension-type headaches
Side Effects
- agranulocytosis
- anaphylactic shock
- anaphylactoid reactions
- anxiety
- aplastic anemia
- azotemia
- confusion
- constipation
- depression
- diarrhea
- disseminated intravascular coagulation (DIC)
- dizziness
- drowsiness
- erythema multiforme
- erythema nodosum
- esophagitis
- excitability
- flatulence
- gastritis
- GI bleeding
- hearing loss
- hemolytic anemia
- hepatic encephalopathy
- hepatic necrosis
- hyperbilirubinemia
- hypertension
- hyperuricemia
- hypoprothrombinemia
- insomnia
- jaundice
- lethargy
- leukopenia
- maculopapular rash
- metabolic acidosis
- nausea
- palpitations
- pancytopenia
- polyuria
- proteinuria
- pruritus
- purpura
- respiratory depression
- Reye’s syndrome
- sinus tachycardia
- thrombocytopenia
- tinnitus
- tolerance
- toxic epidermal necrolysis
- tremor
- vomiting
Monitoring Parameters
- laboratory monitoring not necessary
Contraindications
- abrupt discontinuation
- acid/base imbalance
- acute bronchospasm
- acute myocardial infarction
- agranulocytosis
- alcoholism
- anemia
- angina
- angioedema
- anticoagulant therapy
- ascites
- asthma
- barbiturate hypersensitivity
- bleeding
- bone marrow suppression
- breast-feeding
- carbamazepine hypersensitivity
- cardiac arrhythmias
- cardiac disease
- children
- chronic obstructive pulmonary disease (COPD)
- CNS depression
- coadministration with other CNS depressants
- coagulopathy
- dehydration
- depression
- diabetes mellitus
- driving or operating machinery
- esophagitis
- G6PD deficiency
- gastritis
- geriatric
- GI bleeding
- gout
- heart failure
- hematological disease
- hemophilia
- hepatic disease
- hepatic encephalopathy
- hepatitis
- hydantoin hypersensitivity
- hypertension
- hypoprothrombinemia
- hypotension
- hypothyroidism
- hypovolemia
- immunosuppression
- infants
- infection
- influenza
- labor
- mental status changes
- metabolic acidosis
- metabolic alkalosis
- nasal polyps
- neonates
- neutropenia
- NSAID hypersensitivity
- obstetric delivery
- pain
- peptic ulcer disease
- porphyria
- pregnancy
- prostatic hypertrophy
- pulmonary disease
- renal disease
- renal failure
- renal impairment
- respiratory acidosis
- respiratory alkalosis
- respiratory depression
- Reye’s syndrome
- salicylate hypersensitivity
- sleep apnea
- sodium restriction
- status asthmaticus
- substance abuse
- suicidal ideation
- surgery
- systemic lupus erythematosus (SLE)
- tartrazine dye hypersensitivity
- thrombocytopenia
- thrombolytic therapy
- thrombotic thrombocytopenic purpura (TTP)
- thyroid disease
- tobacco smoking
- urethral stricture
- urticaria
- varicella
- viral infection
- vitamin K deficiency
- von Willebrand’s disease
Interactions
- Abciximab
- Abemaciclib
- Acetaminophen
- Acetaminophen; Aspirin, ASA; Caffeine
- Acetaminophen; Butalbital
- Acetaminophen; Butalbital; Caffeine
- Acetaminophen; Butalbital; Caffeine; Codeine
- Acetaminophen; Caffeine
- Acetaminophen; Caffeine; Dihydrocodeine
- Acetaminophen; Caffeine; Magnesium Salicylate; Phenyltoloxamine
- Acetaminophen; Caffeine; Phenyltoloxamine; Salicylamide
- Acetaminophen; Chlorpheniramine; Dextromethorphan; Phenylephrine
- Acetaminophen; Chlorpheniramine; Dextromethorphan; Pseudoephedrine
- Acetaminophen; Chlorpheniramine; Phenylephrine; Phenyltoloxamine
- Acetaminophen; Codeine
- Acetaminophen; Dextromethorphan
- Acetaminophen; Dextromethorphan; Doxylamine
- Acetaminophen; Dextromethorphan; Guaifenesin; Phenylephrine
- Acetaminophen; Dextromethorphan; Phenylephrine
- Acetaminophen; Dextromethorphan; Pseudoephedrine
- Acetaminophen; Dichloralphenazone; Isometheptene
- Acetaminophen; Diphenhydramine
- Acetaminophen; Guaifenesin; Phenylephrine
- Acetaminophen; Hydrocodone
- Acetaminophen; Oxycodone
- Acetaminophen; Pentazocine
- Acetaminophen; Propoxyphene
- Acetaminophen; Pseudoephedrine
- Acetaminophen; Tramadol
- Acetazolamide
- Acetohexamide
- Acidifying Agents
- Aclidinium; Formoterol
- Acrivastine; Pseudoephedrine
- Adenosine
- Ado-Trastuzumab emtansine
- Albuterol
- Albuterol; Ipratropium
- Aldesleukin, IL-2
- Alfentanil
- Aliskiren; Amlodipine
- Aliskiren; Amlodipine; Hydrochlorothiazide, HCTZ
- Aliskiren; Hydrochlorothiazide, HCTZ
- Alkalinizing Agents
- Alogliptin
- Alogliptin; Metformin
- Alogliptin; Pioglitazone
- Alpha-glucosidase Inhibitors
- Alprazolam
- Altretamine
- Amantadine
- Amiloride
- Amiloride; Hydrochlorothiazide, HCTZ
- Aminoglycosides
- Aminosalicylate sodium, Aminosalicylic acid
- Amiodarone
- Amitriptyline; Chlordiazepoxide
- Amlodipine
- Amlodipine; Atorvastatin
- Amlodipine; Benazepril
- Amlodipine; Celecoxib
- Amlodipine; Hydrochlorothiazide, HCTZ; Olmesartan
- Amlodipine; Hydrochlorothiazide, HCTZ; Valsartan
- Amlodipine; Olmesartan
- Amlodipine; Telmisartan
- Amlodipine; Valsartan
- Amobarbital
- Amoxapine
- Amoxicillin
- Amoxicillin; Clarithromycin; Lansoprazole
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- Buspirone
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- Carbetapentane; Guaifenesin; Phenylephrine
- Carbetapentane; Phenylephrine
- Carbetapentane; Phenylephrine; Pyrilamine
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- Carbetapentane; Pyrilamine
- Carbidopa; Levodopa; Entacapone
- Carbinoxamine
- Carbinoxamine; Dextromethorphan; Pseudoephedrine
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- Carbinoxamine; Hydrocodone; Pseudoephedrine
- Carbinoxamine; Phenylephrine
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- Cariprazine
- Cefixime
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- Cevimeline
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- Chlorothiazide
- Chlorpheniramine
- Chlorpheniramine; Codeine
- Chlorpheniramine; Dextromethorphan
- Chlorpheniramine; Dextromethorphan; Phenylephrine
- Chlorpheniramine; Dihydrocodeine; Phenylephrine
- Chlorpheniramine; Dihydrocodeine; Pseudoephedrine
- Chlorpheniramine; Guaifenesin; Hydrocodone; Pseudoephedrine
- Chlorpheniramine; Hydrocodone
- Chlorpheniramine; Hydrocodone; Phenylephrine
- Chlorpheniramine; Hydrocodone; Pseudoephedrine
- Chlorpheniramine; Phenylephrine
- Chlorpheniramine; Pseudoephedrine
- Chlorpropamide
- Chlorthalidone
- Chlorthalidone; Clonidine
- Choline Salicylate; Magnesium Salicylate
- Cidofovir
- Cilostazol
- Cimetidine
- Cinacalcet
- Ciprofloxacin
- Citalopram
- Citric Acid; Potassium Citrate
- Citric Acid; Potassium Citrate; Sodium Citrate
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- Clemastine
- Clobazam
- Clomipramine
- Clonazepam
- Clopidogrel
- Clorazepate
- Clozapine
- Cobimetinib
- Codeine
- Codeine; Guaifenesin
- Codeine; Phenylephrine; Promethazine
- Codeine; Promethazine
- Colchicine; Probenecid
- Colistimethate, Colistin, Polymyxin E
- Collagenase
- COMT inhibitors
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- Conjugated Estrogens; Bazedoxifene
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- Dalteparin
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- Dapagliflozin; Metformin
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- Darifenacin
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- Dasabuvir; Ombitasvir; Paritaprevir; Ritonavir
- Deferasirox
- Defibrotide
- Deflazacort
- Delavirdine
- Desloratadine; Pseudoephedrine
- Deutetrabenazine
- Dexamethasone
- Dexchlorpheniramine
- Dexchlorpheniramine; Dextromethorphan; Pseudoephedrine
- Dexlansoprazole
- Dexmedetomidine
- Dexmethylphenidate
- Dextroamphetamine
- Dextromethorphan; Diphenhydramine; Phenylephrine
- Dextromethorphan; Guaifenesin; Phenylephrine
- Dextromethorphan; Guaifenesin; Pseudoephedrine
- Dextromethorphan; Quinidine
- Diazepam
- Dichlorphenamide
- Diclofenac
- Diclofenac; Misoprostol
- Dicloxacillin
- Dienogest; Estradiol valerate
- Diethylpropion
- Diethylstilbestrol, DES
- Diflunisal
- Dihydrocodeine; Guaifenesin; Pseudoephedrine
- Diltiazem
- Dimenhydrinate
- Diphenhydramine
- Diphenhydramine; Hydrocodone; Phenylephrine
- Diphenhydramine; Ibuprofen
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- Dipyridamole
- Disopyramide
- Disulfiram
- Dobutamine
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- Doxylamine; Pyridoxine
- Dronabinol
- Dronedarone
- Droperidol
- Drospirenone; Estradiol
- Drospirenone; Ethinyl Estradiol
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- Eltrombopag
- Elvitegravir; Cobicistat; Emtricitabine; Tenofovir Disoproxil Fumarate
- Empagliflozin
- Empagliflozin; Linagliptin
- Empagliflozin; Linagliptin; Metformin
- Empagliflozin; Metformin
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- Emtricitabine; Rilpivirine; Tenofovir disoproxil fumarate
- Emtricitabine; Tenofovir disoproxil fumarate
- Enalapril, Enalaprilat
- Enalapril; Felodipine
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- Ethinyl Estradiol; Norethindrone Acetate
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- Phenothiazines
- Phentermine
- Phentermine; Topiramate
- Phenylephrine
- Phenylephrine; Promethazine
- Phenytoin
- Phosphorated Carbohydrate Solution
- Phosphorus
- Photosensitizing agents (topical)
- Pimavanserin
- Pioglitazone
- Piperacillin
- Piperacillin; Tazobactam
- Pirbuterol
- Piroxicam
- Pneumococcal Vaccine, Polyvalent
- Polymyxins
- Pomalidomide
- Potassium Bicarbonate
- Potassium Chloride
- Potassium Citrate
- Potassium Phosphate
- Potassium Phosphate; Sodium Phosphate
- Pralidoxime
- Pramipexole
- Pramlintide
- Prasterone, Dehydroepiandrosterone, DHEA (Dietary Supplements)
- Prasterone, Dehydroepiandrosterone, DHEA (FDA-approved)
- Prasugrel
- Prednisolone
- Prednisone
- Pregabalin
- Prilocaine; Epinephrine
- Primidone
- Probenecid
- Procarbazine
- Progestins
- Pseudoephedrine
- Psyllium
- Quazepam
- Quetiapine
- Quinapril
- Quinidine
- Quinine
- Rabeprazole
- Racepinephrine
- Ramelteon
- Ramipril
- Ranolazine
- Rasagiline
- Red Yeast Rice
- Regadenoson
- Remifentanil
- Repaglinide
- Reserpine
- Rifampin
- Rifapentine
- Rilpivirine
- Riluzole
- Rimegepant
- Risperidone
- Ritodrine
- Ritonavir
- Rituximab; Hyaluronidase
- Rivaroxaban
- Roflumilast
- Romidepsin
- Ropinirole
- Rosiglitazone
- Rotigotine
- Rucaparib
- Safinamide
- Salicylates
- Salicylic Acid
- Salmeterol
- Salsalate
- Saquinavir
- Saxagliptin
- Scopolamine
- Secobarbital
- Segesterone Acetate; Ethinyl Estradiol
- Selective serotonin reuptake inhibitors
- Selegiline
- Selumetinib
- Serotonin norepinephrine reuptake inhibitors
- Sertraline
- Sibutramine
- Sildenafil
- Simvastatin
- Simvastatin; Sitagliptin
- Siponimod
- Sirolimus
- Sitagliptin
- Skeletal Muscle Relaxants
- Sodium Bicarbonate
- Sodium Hyaluronate, Hyaluronic Acid
- Sodium Lactate
- Sodium Oxybate
- Sodium Thiosulfate; Salicylic Acid
- Solifenacin
- Solriamfetol
- Spironolactone
- St. John’s Wort, Hypericum perforatum
- Sufentanil
- Sulfinpyrazone
- Sulfonamides
- Sulfonylureas
- Sulindac
- Sunitinib
- Suvorexant
- Tacrolimus
- Tapentadol
- Tasimelteon
- Tazemetostat
- Telavancin
- Temazepam
- Tenofovir Alafenamide
- Tenofovir, PMPA
- Terbinafine
- Terbutaline
- Teriflunomide
- Tetrabenazine
- Thalidomide
- Theophylline, Aminophylline
- Thiabendazole
- Thiazide diuretics
- Thiazolidinediones
- Thiopental
- Thiothixene
- Thrombin Inhibitors
- Thrombolytic Agents
- Thyroid hormones
- Ticagrelor
- Ticarcillin
- Ticarcillin; Clavulanic Acid
- Ticlopidine
- Tinzaparin
- Tiotropium; Olodaterol
- Tipranavir
- Tirofiban
- Tizanidine
- tobacco
- Tolazamide
- Tolbutamide
- Tolcapone
- Tolmetin
- Tolterodine
- Topiramate
- Torsemide
- Tramadol
- Trandolapril
- Trandolapril; Verapamil
- Tranylcypromine
- Trastuzumab; Hyaluronidase
- Trazodone
- Treprostinil
- Tretinoin, ATRA
- Triamcinolone
- Triamterene
- Triazolam
- Tricyclic antidepressants
- Trimethobenzamide
- Trimetrexate
- Triprolidine
- Tromethamine
- Ubrogepant
- Ulipristal
- Umeclidinium; Vilanterol
- Valbenazine
- Valerian, Valeriana officinalis
- Valproic Acid, Divalproex Sodium
- Vancomycin
- Varicella-Zoster Virus Vaccine, Live
- Verapamil
- Verteporfin
- Vigabatrin
- Vilazodone
- Vincristine
- Vincristine Liposomal
- Vorapaxar
- Voriconazole
- Vortioxetine
- Voxelotor
- Warfarin
- Yohimbine
- Zafirlukast
- Zaleplon
- Zanubrutinib
- Ziconotide
- Zileuton
- Ziprasidone
- Zolpidem
- Zonisamide