Albiglutide

Albiglutide Brand Name– Tanzeum

What is Albiglutide

Albiglutide is a synthetic glucagon-like peptide-1 receptor agonist (GLP-1 RA) and belongs to a class of antidiabetic agents called incretin mimetics. Incretins are endogenous compounds, including glucagon-like peptide-1 (GLP-1), that improve glycemic control once released into the circulation via the gut.

Albiglutide subcutaneous injection is given just once weekly and is used as an adjunct to diet and exercise to improve glycemic control in adults with type 2 diabetes mellitus (DM).

As with other agents in this class, albiglutide is not recommended as first-line therapy for patients who have inadequate glycemic control on diet and exercise because of the boxed warning regarding rodent C-cell tumor findings and the uncertain relevance to humans.

Indications

  • type 2 diabetes mellitus

For the treatment of type 2 diabetes mellitus in combination with diet and exercise

Side Effects

  1. angioedema
  2. antibody formation
  3. arthralgia
  4. atrial fibrillation
  5. atrial flutter
  6. back pain
  7. constipation
  8. cough
  9. dehydration
  10. diarrhea
  11. dyspepsia
  12. dyspnea
  13. elevated hepatic enzymes
  14. erythema
  15. gastroesophageal reflux
  16. hematoma
  17. hypoglycemia
  18. infection
  19. influenza
  20. injection site reaction
  21. nausea
  22. new primary malignancy
  23. pancreatitis
  24. pruritus
  25. rash
  26. renal failure (unspecified)
  27. sinusitis
  28. vomiting

Monitoring Parameters

  • blood glucose
  • glycosylated hemoglobin A1c (HbA1c)

Contraindications

  • breast-feeding
  • burns
  • children
  • colitis
  • Crohn’s disease
  • dehydration
  • diabetic ketoacidosis
  • diarrhea
  • fever
  • gastroparesis
  • geriatric
  • GI bleeding
  • GI disease
  • GI obstruction
  • GI perforation
  • history of angioedema
  • hypoglycemia
  • ileus
  • infants
  • infection
  • inflammatory bowel disease
  • medullary thyroid carcinoma (MTC)
  • multiple endocrine neoplasia syndrome type 2 (MEN 2)
  • neonates
  • pancreatitis
  • pregnancy
  • pseudomembranous colitis
  • renal failure
  • renal impairment
  • serious hypersensitivity reactions or anaphylaxis
  • surgery
  • thyroid C-cell tumors
  • thyroid cancer
  • thyroid disease
  • tobacco smoking
  • trauma
  • type 1 diabetes mellitus
  • ulcerative colitis
  • vomiting

Interactions

  • Acetaminophen; Aspirin, ASA; Caffeine
  • Acetaminophen; Caffeine; Magnesium Salicylate; Phenyltoloxamine
  • Acetaminophen; Caffeine; Phenyltoloxamine; Salicylamide
  • Acetazolamide
  • Aliskiren; Valsartan
  • Aminosalicylate sodium, Aminosalicylic acid
  • Amlodipine; Benazepril
  • Amlodipine; Hydrochlorothiazide, HCTZ; Olmesartan
  • Amlodipine; Hydrochlorothiazide, HCTZ; Valsartan
  • Amlodipine; Olmesartan
  • Amlodipine; Telmisartan
  • Amlodipine; Valsartan
  • Amoxicillin; Clarithromycin; Lansoprazole
  • Amoxicillin; Clarithromycin; Omeprazole
  • Amprenavir
  • Androgens
  • Angiotensin II receptor antagonists
  • Angiotensin-converting enzyme inhibitors
  • Aspirin, ASA
  • Aspirin, ASA; Butalbital; Caffeine
  • Aspirin, ASA; Butalbital; Caffeine; Codeine
  • Aspirin, ASA; Caffeine; Dihydrocodeine
  • Aspirin, ASA; Caffeine; Orphenadrine
  • Aspirin, ASA; Carisoprodol
  • Aspirin, ASA; Carisoprodol; Codeine
  • Aspirin, ASA; Citric Acid; Sodium Bicarbonate
  • Aspirin, ASA; Dipyridamole
  • Aspirin, ASA; Omeprazole
  • Aspirin, ASA; Oxycodone
  • Aspirin, ASA; Pravastatin
  • Atazanavir
  • Atazanavir; Cobicistat
  • Atropine; Benzoic Acid; Hyoscyamine; Methenamine; Methylene Blue; Phenyl Salicylate
  • atypical antipsychotic
  • Azilsartan
  • Azilsartan; Chlorthalidone
  • Benazepril
  • Benazepril; Hydrochlorothiazide, HCTZ
  • Benzoic Acid; Hyoscyamine; Methenamine; Methylene Blue; Phenyl Salicylate
  • Beta-blockers
  • Bismuth Subsalicylate
  • Bismuth Subsalicylate; Metronidazole; Tetracycline
  • Bortezomib
  • Candesartan
  • Candesartan; Hydrochlorothiazide, HCTZ
  • Captopril
  • Captopril; Hydrochlorothiazide, HCTZ
  • Carbonic anhydrase inhibitors
  • Chloroquine
  • Chlorpromazine
  • Chlorthalidone; Clonidine
  • Choline Salicylate; Magnesium Salicylate
  • Chromium
  • Clarithromycin
  • Clonidine
  • Codeine; Phenylephrine; Promethazine
  • Codeine; Promethazine
  • Conjugated Estrogens; Medroxyprogesterone
  • Corticosteroids
  • Cyclosporine
  • Daclatasvir
  • Danazol
  • Darunavir
  • Darunavir; Cobicistat
  • Darunavir; Cobicistat; Emtricitabine; Tenofovir alafenamide
  • Dasabuvir; Ombitasvir; Paritaprevir; Ritonavir
  • Dasabuvir; Ombitasvir; Paritaprevir; Ritonavir
  • Dextromethorphan; Promethazine
  • Diazoxide
  • Dienogest; Estradiol valerate
  • Disopyramide
  • Drospirenone
  • Drospirenone; Estradiol
  • Drospirenone; Ethinyl Estradiol
  • Drospirenone; Ethinyl Estradiol; Levomefolate
  • Elagolix; Estradiol; Norethindrone acetate
  • Elbasvir; Grazoprevir
  • Enalapril, Enalaprilat
  • Enalapril; Felodipine
  • Enalapril; Hydrochlorothiazide, HCTZ
  • Eprosartan
  • Eprosartan; Hydrochlorothiazide, HCTZ
  • Esterified Estrogens; Methyltestosterone
  • Estradiol Cypionate; Medroxyprogesterone
  • Estradiol; Levonorgestrel
  • Estradiol; Norethindrone
  • Estradiol; Norgestimate
  • Estradiol; Progesterone
  • Estrogens
  • Ethanol
  • Ethinyl Estradiol; Desogestrel
  • Ethinyl Estradiol; Ethynodiol Diacetate
  • Ethinyl Estradiol; Etonogestrel
  • Ethinyl Estradiol; Levonorgestrel
  • Ethinyl Estradiol; Levonorgestrel; Ferrous bisglycinate
  • Ethinyl Estradiol; Levonorgestrel; Folic Acid; Levomefolate
  • Ethinyl Estradiol; Norelgestromin
  • Ethinyl Estradiol; Norethindrone
  • Ethinyl Estradiol; Norethindrone Acetate
  • Ethinyl Estradiol; Norethindrone Acetate; Ferrous fumarate
  • Ethinyl Estradiol; Norethindrone; Ferrous fumarate
  • Ethinyl Estradiol; Norgestimate
  • Ethinyl Estradiol; Norgestrel
  • Ethotoin
  • Etonogestrel
  • Fibric acid derivatives
  • Fluoxetine
  • Fluoxetine; Olanzapine
  • Fluoxymesterone
  • Fluphenazine
  • Fosamprenavir
  • Fosinopril
  • Fosinopril; Hydrochlorothiazide, HCTZ
  • Fosphenytoin
  • Garlic, Allium sativum
  • Glecaprevir; Pibrentasvir
  • Green Tea
  • Hydrochlorothiazide, HCTZ; Irbesartan
  • Hydrochlorothiazide, HCTZ; Lisinopril
  • Hydrochlorothiazide, HCTZ; Losartan
  • Hydrochlorothiazide, HCTZ; Moexipril
  • Hydrochlorothiazide, HCTZ; Olmesartan
  • Hydrochlorothiazide, HCTZ; Quinapril
  • Hydrochlorothiazide, HCTZ; Telmisartan
  • Hydrochlorothiazide, HCTZ; Triamterene
  • Hydrochlorothiazide, HCTZ; Valsartan
  • Hydroxychloroquine
  • Hydroxyprogesterone
  • Hyoscyamine; Methenamine; Methylene Blue; Phenyl Salicylate; Sodium Biphosphate
  • Indapamide
  • Indinavir
  • Insulin Detemir
  • Irbesartan
  • Isocarboxazid
  • Lanreotide
  • Ledipasvir; Sofosbuvir
  • Leuprolide; Norethindrone
  • Levonorgestrel
  • Levothyroxine
  • Levothyroxine; Liothyronine (Porcine)
  • Levothyroxine; Liothyronine (Synthetic)
  • Linezolid
  • Liothyronine
  • Lisinopril
  • Lithium
  • Lomefloxacin
  • Loop diuretics
  • Lopinavir; Ritonavir
  • Lorcaserin
  • Losartan
  • Lovastatin; Niacin
  • Magnesium Salicylate
  • Mecasermin rinfabate
  • Mecasermin, Recombinant, rh-IGF-1
  • Medroxyprogesterone
  • Meperidine; Promethazine
  • Mesoridazine
  • Mestranol; Norethindrone
  • Methazolamide
  • Methyltestosterone
  • Metyrapone
  • Moexipril
  • Monoamine oxidase inhibitors
  • Nandrolone Decanoate
  • Nebivolol; Valsartan
  • Nelfinavir
  • Niacin, Niacinamide
  • Niacin; Simvastatin
  • Nicotine
  • Norethindrone
  • Norgestrel
  • Octreotide
  • Olmesartan
  • Ombitasvir; Paritaprevir; Ritonavir
  • Orlistat
  • Oxandrolone
  • Oxymetholone
  • Pasireotide
  • Pegvisomant
  • Pentamidine
  • Pentoxifylline
  • Perindopril
  • Perindopril; Amlodipine
  • Perphenazine
  • Perphenazine; Amitriptyline
  • Phenelzine
  • Phenothiazines
  • Phenylephrine; Promethazine
  • Phenytoin
  • Prasterone, Dehydroepiandrosterone, DHEA (Dietary Supplements)
  • Prasterone, Dehydroepiandrosterone, DHEA (FDA-approved)
  • Prochlorperazine
  • Progesterone
  • Progestins
  • Promethazine
  • Protease inhibitors
  • Quinapril
  • Quinolones
  • Ramipril
  • Reserpine
  • Ritonavir
  • Sacubitril; Valsartan
  • Salicylates
  • Salsalate
  • Saquinavir
  • Segesterone Acetate; Ethinyl Estradiol
  • Selegiline
  • Sofosbuvir
  • Sofosbuvir; Velpatasvir
  • Sofosbuvir; Velpatasvir; Voxilaprevir
  • Somatropin, rh-GH
  • Sparfloxacin
  • Sulfonamides
  • Sympathomimetics
  • Tacrolimus
  • Tegaserod
  • Telmisartan
  • Testolactone
  • Testosterone
  • Thiazide diuretics
  • Thiethylperazine
  • Thioridazine
  • Thyroid hormones
  • Tipranavir
  • tobacco
  • Trandolapril
  • Trandolapril; Verapamil
  • Tranylcypromine
  • Triamterene
  • Trifluoperazine
  • Valsartan
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