What are p38 kinase inhibitors?
The p38 mitogen-activated protein kinases are responsive to stress stimuli, such as cytokines, resulting in inflammation. Inhibition of these kinases is antiinflammatory. They have potential utility in autoimmune disease and inflammatory states; however, clinical trials to date have not been successful. Inhibition may result in prolonged QTc interval and will be contraindicated in patients at risk for arrhythmias.
Related Posts
-
mtor inhibitorsWhat are mtor inhibitors? mTOR inhibitors block the mTOR and thus prevent cytokine signals from…
-
-
Main drugs for maintenance therapyWhat are the main drugs used for maintenance therapy? 1. Calcineurin inhibitors (CNI): tacrolimus, cyclosporine2. Anti-metabolites: azathioprine,…
-
Calcineurin Inhibitors (CNIs)What are Calcineurin Inhibitors (CNIs)? Calcineurin Inhibitors remain a cornerstone of immunosuppressive regiments in kidney…