Bumetanide

Bumetanide Brand Name– Bumex

What is Bumetanide

Bumetanide is a sulfonamide-derived loop diuretic used in the management of edema associated with congestive heart failure, cirrhosis, and renal disease such as nephrotic syndrome.

It is structurally related to furosemide, but its diuretic potency is about 40 times greater.

Bumetanide may be particularly useful in patients who are unresponsive to other diuretics or who have severe renal impairment and require large doses of loop diuretics.

Bumetanide was approved by the FDA in 1983.

Indications

  1. ascites
  2. edema
  3. heart failure
  4. hypercalcemia
  5. hypertension
  6. nephrotic syndrome
  7. oliguria

For the treatment of peripheral edema or edema associated with heart failure or nephrotic syndrome

Monitoring Parameters

  • blood glucose
  • serum creatinine/BUN
  • serum electrolytes
  • serum uric acid

Contraindications

  • acid/base imbalance
  • acute myocardial infarction
  • anuria
  • breast-feeding
  • children
  • dehydration
  • diabetes mellitus
  • diarrhea
  • electrolyte imbalance
  • geriatric
  • gout
  • hearing impairment
  • heart failure
  • hepatic disease
  • hepatic encephalopathy
  • hyperglycemia
  • hyperuricemia
  • hypocalcemia
  • hypochloremia
  • hypokalemia
  • hypomagnesemia
  • hyponatremia
  • hypotension
  • hypovolemia
  • infants
  • jaundice
  • metabolic alkalosis
  • neonates
  • oliguria
  • orthostatic hypotension
  • pancreatitis
  • pregnancy
  • renal disease
  • renal failure
  • renal impairment
  • sulfonamide hypersensitivity
  • sympathectomy
  • syncope
  • thiazide diuretic hypersensitivity
  • tinnitus
  • ventricular arrhythmias

Interactions

  • Acarbose
  • Acetaminophen; Butalbital; Caffeine; Codeine
  • Acetaminophen; Chlorpheniramine; Dextromethorphan; Phenylephrine
  • Acetaminophen; Chlorpheniramine; Dextromethorphan; Pseudoephedrine
  • Acetaminophen; Chlorpheniramine; Phenylephrine; Phenyltoloxamine
  • Acetaminophen; Codeine
  • Acetaminophen; Dextromethorphan; Guaifenesin; Phenylephrine
  • Acetaminophen; Dextromethorphan; Phenylephrine
  • Acetaminophen; Dextromethorphan; Pseudoephedrine
  • Acetaminophen; Dichloralphenazone; Isometheptene
  • Acetaminophen; Guaifenesin; Phenylephrine
  • Acetaminophen; Hydrocodone
  • Acetaminophen; Oxycodone
  • Acetaminophen; Pentazocine
  • Acetaminophen; Pseudoephedrine
  • Acetaminophen; Tramadol
  • Acetazolamide
  • Acrivastine; Pseudoephedrine
  • Albiglutide
  • Alemtuzumab
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  • Alfentanil
  • Aliskiren
  • Aliskiren; Amlodipine
  • Aliskiren; Amlodipine; Hydrochlorothiazide, HCTZ
  • Aliskiren; Hydrochlorothiazide, HCTZ
  • Aliskiren; Valsartan
  • Alogliptin
  • Alogliptin; Metformin
  • Alogliptin; Pioglitazone
  • Alpha-glucosidase Inhibitors
  • Alprostadil
  • Aluminum Hydroxide; Magnesium Hydroxide
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  • Amiloride; Hydrochlorothiazide, HCTZ
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  • Amiodarone
  • Amlodipine; Benazepril
  • Amlodipine; Celecoxib
  • Amlodipine; Hydrochlorothiazide, HCTZ; Olmesartan
  • Amlodipine; Hydrochlorothiazide, HCTZ; Valsartan
  • Amlodipine; Olmesartan
  • Amlodipine; Telmisartan
  • Amlodipine; Valsartan
  • Amobarbital
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  • Amoxicillin; Clarithromycin; Omeprazole
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  • Enalapril; Hydrochlorothiazide, HCTZ
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  • Eprosartan; Hydrochlorothiazide, HCTZ
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  • Esomeprazole; Naproxen
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  • Fospropofol
  • Gallium Ga 68 Dotatate
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  • Granisetron
  • Guaifenesin; Hydrocodone
  • Guaifenesin; Hydrocodone; Pseudoephedrine
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  • Halothane
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