Aminosalicylate sodium and Aminosalicylic acid Brand Name– PASER
What is Aminosalicylate sodium and Aminosalicylic acid
Aminosalicylate sodium and aminosalicylic acid are analogs of aminobenzoic acid (PABA) and are used orally as antituberculosis agents.
They are administered as adjunct agents in combination with at least one other antituberculosis agent.
Aminosalicylate sodium and aminosalicylic acid are usually reserved as last-line agents secondary to effectiveness.
Aminosalicylate sodium was approved prior to 1982 and aminosalicylic acid was approved in 1994.
Indications
- aminosalicylic acid desensitization
- Mycobacterium tuberculosis
- tuberculosis infection
Side Effects
- abdominal pain
- agranulocytosis
- crystalluria
- diarrhea
- encephalopathy
- exfoliative dermatitis
- fever
- hemolytic anemia
- hepatitis
- hypoglycemia
- jaundice
- leukopenia
- nausea
- optic neuritis
- pericarditis
- thrombocytopenia
- vasculitis
- vomiting
Monitoring Parameters
- serum creatinine/BUN
Contraindications
- breast-feeding
- hepatic disease
- hepatitis
- jaundice
- malabsorption syndrome
- pregnancy
- renal disease
- renal failure
- vitamin B12 deficiency
Interactions
- Acetazolamide
- Aliskiren; Amlodipine; Hydrochlorothiazide, HCTZ
- Aliskiren; Hydrochlorothiazide, HCTZ
- Alogliptin
- Alogliptin; Metformin
- Alogliptin; Pioglitazone
- Alpha-glucosidase Inhibitors
- Amiloride
- Amiloride; Hydrochlorothiazide, HCTZ
- Aminoglycosides
- Amlodipine; Benazepril
- Amlodipine; Hydrochlorothiazide, HCTZ; Olmesartan
- Amlodipine; Hydrochlorothiazide, HCTZ; Valsartan
- Amphotericin B
- Amphotericin B cholesteryl sulfate complex (ABCD)
- Amphotericin B lipid complex (ABLC)
- Amphotericin B liposomal (LAmB)
- Angiotensin-converting enzyme inhibitors
- Antithrombin III
- Antithymocyte Globulin
- Apixaban
- Ardeparin
- Articaine; Epinephrine
- Atenolol; Chlorthalidone
- Azilsartan; Chlorthalidone
- Bacitracin
- Barbiturates
- Benazepril
- Benazepril; Hydrochlorothiazide, HCTZ
- Bendroflumethiazide; Nadolol
- Bisoprolol; Hydrochlorothiazide, HCTZ
- Bromocriptine
- Bumetanide
- Bupivacaine
- Bupivacaine Liposomal
- Bupivacaine; Lidocaine
- Calcium Carbonate
- Calcium Carbonate; Magnesium Hydroxide
- Calcium Carbonate; Risedronate
- Calcium Carbonate; Simethicone
- Canagliflozin
- Canagliflozin; Metformin
- Candesartan; Hydrochlorothiazide, HCTZ
- Capreomycin
- Captopril
- Captopril; Hydrochlorothiazide, HCTZ
- Cefixime
- Cefotetan
- Chloroprocaine
- Chlorothiazide
- Chlorthalidone
- Chlorthalidone; Clonidine
- Citric Acid; Potassium Citrate
- Citric Acid; Potassium Citrate; Sodium Citrate
- Colchicine; Probenecid
- Colistimethate, Colistin, Polymyxin E
- Corticosteroids
- Cyclosporine
- Dabigatran
- Dalteparin
- Dapagliflozin
- Dapagliflozin; Metformin
- Dapagliflozin; Saxagliptin
- Daratumumab; Hyaluronidase
- Deferasirox
- Diclofenac
- Diclofenac; Misoprostol
- Diflunisal
- Diphenhydramine; Ibuprofen
- Diphenhydramine; Naproxen
- Doravirine; Lamivudine; Tenofovir disoproxil fumarate
- Drotrecogin Alfa
- Edoxaban
- Efavirenz; Emtricitabine; Tenofovir
- Efavirenz; Lamivudine; Tenofovir Disoproxil Fumarate
- Elvitegravir; Cobicistat; Emtricitabine; Tenofovir Disoproxil Fumarate
- Empagliflozin
- Empagliflozin; Linagliptin
- Empagliflozin; Linagliptin; Metformin
- Empagliflozin; Metformin
- Emtricitabine; Rilpivirine; Tenofovir disoproxil fumarate
- Emtricitabine; Tenofovir disoproxil fumarate
- Enalapril, Enalaprilat
- Enalapril; Felodipine
- Enalapril; Hydrochlorothiazide, HCTZ
- Enoxaparin
- Eprosartan; Hydrochlorothiazide, HCTZ
- Ertugliflozin; Metformin
- Ertugliflozin; Sitagliptin
- Esomeprazole; Naproxen
- Ethacrynic Acid
- Ethambutol
- Ethanol
- Ethionamide
- Ethotoin
- Etodolac
- Famotidine; Ibuprofen
- Fenoprofen
- Flurbiprofen
- Fondaparinux
- Foscarnet
- Fosinopril
- Fosinopril; Hydrochlorothiazide, HCTZ
- Fosphenytoin
- Furosemide
- Gallium Ga 68 Dotatate
- Glimepiride; Pioglitazone
- Glimepiride; Rosiglitazone
- Glipizide; Metformin
- Glyburide; Metformin
- Griseofulvin
- Heparin
- Hyaluronidase
- Hyaluronidase, Recombinant; Immune Globulin
- Hydralazine; Hydrochlorothiazide, HCTZ
- Hydrochlorothiazide, HCTZ
- Hydrochlorothiazide, HCTZ; Irbesartan
- Hydrochlorothiazide, HCTZ; Lisinopril
- Hydrochlorothiazide, HCTZ; Losartan
- Hydrochlorothiazide, HCTZ; Methyldopa
- Hydrochlorothiazide, HCTZ; Metoprolol
- Hydrochlorothiazide, HCTZ; Moexipril
- Hydrochlorothiazide, HCTZ; Olmesartan
- Hydrochlorothiazide, HCTZ; Propranolol
- Hydrochlorothiazide, HCTZ; Quinapril
- Hydrochlorothiazide, HCTZ; Spironolactone
- Hydrochlorothiazide, HCTZ; Telmisartan
- Hydrochlorothiazide, HCTZ; Triamterene
- Hydrochlorothiazide, HCTZ; Valsartan
- Hydrocodone; Ibuprofen
- Ibuprofen
- Ibuprofen; Oxycodone
- Ibuprofen; Pseudoephedrine
- Incretin Mimetics
- Indapamide
- Inotersen
- Insulins
- Isoniazid, INH
- Isoniazid, INH; Pyrazinamide, PZA; Rifampin
- Isoniazid, INH; Rifampin
- Ketoprofen
- Ketorolac
- Lamivudine; Tenofovir Disoproxil Fumarate
- Lansoprazole; Naproxen
- Lidocaine
- Lidocaine; Prilocaine
- Linagliptin
- Linagliptin; Metformin
- Lisinopril
- Loop diuretics
- Low Molecular Weight Heparins
- Macimorelin
- Mannitol
- Measles Virus; Mumps Virus; Rubella Virus; Varicella Virus Vaccine, Live
- Meclofenamate Sodium
- Mefenamic Acid
- Meglitinides
- Meloxicam
- Mepivacaine
- Mepivacaine; Levonordefrin
- Metformin
- Metformin; Pioglitazone
- Metformin; Repaglinide
- Metformin; Rosiglitazone
- Metformin; Saxagliptin
- Metformin; Sitagliptin
- Methazolamide
- Methotrexate
- Methyclothiazide
- Metolazone
- Moexipril
- Mycophenolate
- Nabumetone
- Naproxen
- Naproxen; Pseudoephedrine
- Naproxen; Sumatriptan
- Nateglinide
- Nitazoxanide
- Omeprazole; Amoxicillin; Rifabutin
- Oxaprozin
- Penicillin G Benzathine; Penicillin G Procaine
- Penicillin G Procaine
- Pentosan
- Perindopril
- Perindopril; Amlodipine
- Phentermine; Topiramate
- Phenytoin
- Photosensitizing agents (topical)
- Pioglitazone
- Piroxicam
- Polymyxins
- Potassium Bicarbonate
- Potassium Chloride
- Potassium Citrate
- Pramlintide
- Prilocaine
- Prilocaine; Epinephrine
- Probenecid
- Psyllium
- Pyrazinamide, PZA
- Quinapril
- Ramipril
- Repaglinide
- Rifabutin
- Rifampin
- Rituximab; Hyaluronidase
- Rivaroxaban
- Ropivacaine
- Rosiglitazone
- Salicylic Acid
- Saxagliptin
- Serotonin norepinephrine reuptake inhibitors
- Simvastatin; Sitagliptin
- Sitagliptin
- Sodium Hyaluronate, Hyaluronic Acid
- Sodium Thiosulfate; Salicylic Acid
- Spironolactone
- Sulfinpyrazone
- Sulfonamides
- Sulindac
- Tacrolimus
- Telavancin
- Tenofovir Alafenamide
- Tenofovir, PMPA
- Tetracaine
- Thiazide diuretics
- Thiazolidinediones
- Thrombin Inhibitors
- Thrombolytic Agents
- Tinzaparin
- Tolmetin
- Topiramate
- Torsemide
- Trandolapril
- Trandolapril; Verapamil
- Trastuzumab; Hyaluronidase
- Trazodone
- Treprostinil
- Triamterene
- Valproic Acid, Divalproex Sodium
- Vancomycin
- Varicella-Zoster Virus Vaccine, Live
- Vilazodone
- Vortioxetine