Indinavir

Indinavir Brand Name– Chemet | Crixivan

What is Indinavir

Indinavir is a protease inhibitor approved for use in combination with other antiretroviral medications to treat human immunodeficiency virus (HIV-1) infections.

Concerns about high pill burden (when used without ritonavir) and the potential for nephrolithiasis may limit its use.

Adequate hydration (1.5 liters per 24 hour period) is recommended in all patients treated with indinavir.

Indications

  1. human immunodeficiency virus (HIV)
  2. human immunodeficiency virus (HIV) infection

Side Effects

  1. abdominal pain
  2. alopecia
  3. anaphylactoid reactions
  4. anemia
  5. angina
  6. anorexia
  7. appetite stimulation
  8. arthralgia
  9. asthenia
  10. back pain
  11. bleeding
  12. cough
  13. crystalluria
  14. Cushingoid features
  15. depression
  16. diabetes mellitus
  17. diabetic ketoacidosis
  18. diarrhea
  19. dizziness
  20. drowsiness
  21. dysgeusia
  22. dyspepsia
  23. dysuria
  24. elevated hepatic enzymes
  25. erythema multiforme
  26. fatigue
  27. fever
  28. flank pain
  29. gastroesophageal reflux
  30. GI bleeding
  31. gynecomastia
  32. headache
  33. hematoma
  34. hematuria
  35. hemolytic anemia
  36. hepatic failure
  37. hepatitis
  38. hyperamylasemia
  39. hyperbilirubinemia
  40. hypercholesterolemia
  41. hyperglycemia
  42. hyperlipidemia
  43. hypertriglyceridemia
  44. interstitial nephritis
  45. intracranial bleeding
  46. jaundice
  47. lipodystrophy
  48. malaise
  49. myocardial infarction
  50. nausea
  51. nephrolithiasis
  52. neutropenia
  53. pancreatitis
  54. paresthesias
  55. pruritus
  56. rash
  57. renal tubular obstruction
  58. skin hyperpigmentation
  59. Stevens-Johnson syndrome
  60. thrombocytopenia
  61. urticaria
  62. vasculitis
  63. vomiting
  64. xerosis

Monitoring Parameters

  • blood glucose
  • CBC with differential
  • CD4+ T cell count
  • hepatitis B serology
  • LFTs
  • plasma hepatitis C RNA
  • plasma HIV RNA
  • pregnancy testing
  • serum bilirubin (total and direct)
  • serum cholesterol
  • serum lipid profile
  • urinalysis

Contraindications

  • autoimmune disease
  • breast-feeding
  • children
  • dehydration
  • diabetes mellitus
  • diabetic ketoacidosis
  • Graves’ disease
  • Guillain-Barre syndrome
  • hemophilia
  • hepatic disease
  • hepatitis
  • hepatitis B and HIV coinfection
  • hepatitis C and HIV coinfection
  • human immunodeficiency virus (HIV) infection resistance
  • hypercholesterolemia
  • hyperglycemia
  • hyperlipidemia
  • hypertriglyceridemia
  • immune reconstitution syndrome
  • infants
  • labor
  • neonates
  • nephrolithiasis
  • pancreatitis
  • pregnancy
  • tuberculosis

Interactions

  • Abacavir; Lamivudine, 3TC; Zidovudine, ZDV
  • Abemaciclib
  • Acalabrutinib
  • Acarbose
  • Acetaminophen; Butalbital
  • Acetaminophen; Butalbital; Caffeine
  • Acetaminophen; Butalbital; Caffeine; Codeine
  • Acetaminophen; Caffeine; Dihydrocodeine
  • Acetaminophen; Codeine
  • Acetaminophen; Hydrocodone
  • Acetaminophen; Oxycodone
  • Acetaminophen; Propoxyphene
  • Adefovir
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  • Aldesleukin, IL-2
  • Alfentanil
  • Alfuzosin
  • Aliskiren; Amlodipine
  • Aliskiren; Amlodipine; Hydrochlorothiazide, HCTZ
  • Almotriptan
  • Alogliptin
  • Alogliptin; Metformin
  • Alogliptin; Pioglitazone
  • Alosetron
  • Alpha-glucosidase Inhibitors
  • Alprazolam
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  • Amlodipine; Celecoxib
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  • Amlodipine; Hydrochlorothiazide, HCTZ; Valsartan
  • Amlodipine; Olmesartan
  • Amlodipine; Telmisartan
  • Amlodipine; Valsartan
  • Amobarbital
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  • Aspirin, ASA; Caffeine; Dihydrocodeine
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  • Aspirin, ASA; Omeprazole
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  • food
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  • grapefruit juice
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  • Haloperidol
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