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Ibritumomab Tiuxetan Brand Names- Zevalin for In-111 | Zevalin for Y-90
What is Ibritumomab Tiuxetan
Ibritumomab tiuxetan is a radiotherapeutic monoclonal antibody that binds to the CD20 molecule found on pre B- and mature B-lymphocytes.
It is indicated in combination with rituximab for relapsed or refractory, low-grade or follicular B-cell non-Hodgkin lymphoma (NHL) and previously untreated follicular NHL in patients who achieve a partial or complete response to first-line chemotherapy.
Serious infusion reactions, prolonged and severe cytopenias, and severe cutaneous and mucocutaneous reactions have been reported with ibritumomab tiuxetan therapy.
Indications
- non-Hodgkin’s lymphoma (NHL)
For the treatment of non-Hodgkin’s lymphoma (NHL)
Side Effects
- abdominal pain
- abdominal pain
- acute respiratory distress syndrome (ARDS)
- anemia
- anemia
- angioedema
- anorexia
- antibody formation
- asthenia
- asthenia
- bone marrow suppression
- bronchospasm
- bullous rash
- cough
- cough
- diarrhea
- dizziness
- ecchymosis
- ecchymosis
- epistaxis
- epistaxis
- erythema
- erythema multiforme
- exfoliative dermatitis
- fatigue
- fatigue
- fever
- fever
- hypertension
- hypertension
- hypotension
- hypoxia
- infection
- infection
- influenza
- infusion-related reactions
- leukemia
- leukopenia
- leukopenia
- lymphopenia
- lymphopenia
- myalgia
- myocardial infarction
- nausea
- neutropenia
- neutropenia
- new primary malignancy
- night sweats
- petechiae
- petechiae
- pharyngitis
- pruritus
- rash
- rash
- rhinitis
- sinusitis
- sinusitis
- skin necrosis
- skin ulcer
- Stevens-Johnson syndrome
- thrombocytopenia
- thrombocytopenia
- toxic epidermal necrolysis
- urticaria
- ventricular fibrillation
Monitoring Parameters
- CBC with differential
- platelet count
- pregnancy testing
Contraindications
- accidental exposure
- anticoagulant therapy
- bleeding
- bone marrow suppression
- breast-feeding
- contraception requirements
- extravasation
- infection
- infertility
- infusion-related reactions
- male-mediated teratogenicity
- neutropenia
- new primary malignancy
- pregnancy
- pregnancy testing
- reproductive risk
- serious rash
- thrombocytopenia
- vaccination
Interactions
- Abciximab
- Acetaminophen; Aspirin, ASA; Caffeine
- Acetaminophen; Caffeine; Magnesium Salicylate; Phenyltoloxamine
- Acetaminophen; Chlorpheniramine; Dextromethorphan; Pseudoephedrine
- Acetaminophen; Dextromethorphan; Pseudoephedrine
- Acetaminophen; Pseudoephedrine
- Acrivastine; Pseudoephedrine
- Alendronate; Cholecalciferol
- Aliskiren
- Aliskiren; Amlodipine
- Aliskiren; Amlodipine; Hydrochlorothiazide, HCTZ
- Aliskiren; Hydrochlorothiazide, HCTZ
- Aliskiren; Valsartan
- Alpha interferons
- Alteplase
- Aluminum Hydroxide
- Aluminum Hydroxide; Magnesium Carbonate
- Aluminum Hydroxide; Magnesium Hydroxide
- Aluminum Hydroxide; Magnesium Hydroxide; Simethicone
- Aluminum Hydroxide; Magnesium Trisilicate
- Amiloride
- Amiloride; Hydrochlorothiazide, HCTZ
- Amlodipine; Benazepril
- Amlodipine; Celecoxib
- Amlodipine; Hydrochlorothiazide, HCTZ; Olmesartan
- Amlodipine; Hydrochlorothiazide, HCTZ; Valsartan
- Amlodipine; Olmesartan
- Amlodipine; Telmisartan
- Amlodipine; Valsartan
- Ammonium Chloride
- Amphetamines
- Anagrelide
- Angiotensin II receptor antagonists
- Angiotensin-converting enzyme inhibitors
- Antacids
- Anticholinergics
- Anticoagulants
- Antithrombin III
- Antithymocyte Globulin
- Apixaban
- Argatroban
- Aspirin, ASA
- Aspirin, ASA; Butalbital; Caffeine
- Aspirin, ASA; Butalbital; Caffeine; Codeine
- Aspirin, ASA; Caffeine; Dihydrocodeine
- Aspirin, ASA; Caffeine; Orphenadrine
- Aspirin, ASA; Carisoprodol
- Aspirin, ASA; Carisoprodol; Codeine
- Aspirin, ASA; Citric Acid; Sodium Bicarbonate
- Aspirin, ASA; Dipyridamole
- Aspirin, ASA; Omeprazole
- Aspirin, ASA; Oxycodone
- Aspirin, ASA; Pravastatin
- Atropine
- Atropine; Benzoic Acid; Hyoscyamine; Methenamine; Methylene Blue; Phenyl Salicylate
- Atropine; Difenoxin
- Atropine; Diphenoxylate
- Atropine; Edrophonium
- Atropine; Hyoscyamine; Phenobarbital; Scopolamine
- Azelastine; Fluticasone
- Azilsartan
- Azilsartan; Chlorthalidone
- Beclomethasone
- Belladonna Alkaloids; Ergotamine; Phenobarbital
- Belladonna; Opium
- Benazepril
- Benazepril; Hydrochlorothiazide, HCTZ
- Benzoic Acid; Hyoscyamine; Methenamine; Methylene Blue; Phenyl Salicylate
- Benztropine
- Betamethasone
- Betrixaban
- Bismuth Subsalicylate
- Bismuth Subsalicylate; Metronidazole; Tetracycline
- Bivalirudin
- Brompheniramine; Hydrocodone; Pseudoephedrine
- Brompheniramine; Pseudoephedrine
- Budesonide
- Budesonide; Formoterol
- Burosumab
- Caffeine
- Calcium
- Calcium Carbonate; Magnesium Hydroxide
- Calcium; Vitamin D
- Candesartan
- Candesartan; Hydrochlorothiazide, HCTZ
- Captopril
- Captopril; Hydrochlorothiazide, HCTZ
- Carbetapentane; Guaifenesin; Phenylephrine
- Carbetapentane; Phenylephrine
- Carbetapentane; Pseudoephedrine
- Carbinoxamine; Dextromethorphan; Pseudoephedrine
- Carbinoxamine; Hydrocodone; Pseudoephedrine
- Carbinoxamine; Pseudoephedrine
- Celecoxib
- Cetirizine; Pseudoephedrine
- Chlophedianol; Dexchlorpheniramine; Pseudoephedrine
- Chlordiazepoxide; Clidinium
- Chlorpheniramine; Dihydrocodeine; Pseudoephedrine
- Chlorpheniramine; Guaifenesin; Hydrocodone; Pseudoephedrine
- Chlorpheniramine; Hydrocodone; Pseudoephedrine
- Chlorpheniramine; Pseudoephedrine
- Chlorpropamide
- Choline Salicylate; Magnesium Salicylate
- Ciclesonide
- Cilostazol
- Clopidogrel
- Clozapine
- Colchicine
- Colchicine; Probenecid
- Colestipol
- Corticosteroids
- Cortisone
- Cyclosporine
- Dabigatran
- Dalteparin
- Danaparoid
- Deflazacort
- Desirudin
- Desloratadine; Pseudoephedrine
- Dexamethasone
- Dexchlorpheniramine; Dextromethorphan; Pseudoephedrine
- Dextromethorphan; Guaifenesin; Pseudoephedrine
- Dextromethorphan; Quinidine
- Diazoxide
- Dichlorphenamide
- Diclofenac
- Diclofenac; Misoprostol
- Dicyclomine
- Diflunisal
- Digoxin
- Dihydrocodeine; Guaifenesin; Pseudoephedrine
- Diphenhydramine; Ibuprofen
- Diphenhydramine; Naproxen
- Dipyridamole
- Donepezil; Memantine
- Drospirenone
- Drospirenone; Estradiol
- Drospirenone; Ethinyl Estradiol
- Drospirenone; Ethinyl Estradiol; Levomefolate
- Echinacea
- Edoxaban
- Enalapril, Enalaprilat
- Enalapril; Felodipine
- Enalapril; Hydrochlorothiazide, HCTZ
- Enoxaparin
- Eplerenone
- Eprosartan
- Eprosartan; Hydrochlorothiazide, HCTZ
- Eptifibatide
- Erdafitinib
- Ergocalciferol, Vitamin D2
- Esomeprazole; Naproxen
- Etodolac
- Famotidine; Ibuprofen
- Fenoprofen
- Fexofenadine; Pseudoephedrine
- Filgrastim, G-CSF
- Flavoxate
- Flecainide
- Fludrocortisone
- Flunisolide
- Flurbiprofen
- Fluticasone
- Fluticasone; Salmeterol
- Fluticasone; Umeclidinium; Vilanterol
- Fluticasone; Vilanterol
- Fondaparinux
- food
- Formoterol; Mometasone
- Fosinopril
- Fosinopril; Hydrochlorothiazide, HCTZ
- Glycopyrrolate
- Glycopyrrolate; Formoterol
- Guaifenesin; Hydrocodone; Pseudoephedrine
- Guaifenesin; Pseudoephedrine
- Heparin
- Hetastarch; Dextrose; Electrolytes
- Homatropine; Hydrocodone
- Hydralazine
- Hydralazine; Hydrochlorothiazide, HCTZ
- Hydralazine; Isosorbide Dinitrate, ISDN
- Hydrochlorothiazide, HCTZ; Irbesartan
- Hydrochlorothiazide, HCTZ; Lisinopril
- Hydrochlorothiazide, HCTZ; Losartan
- Hydrochlorothiazide, HCTZ; Methyldopa
- Hydrochlorothiazide, HCTZ; Moexipril
- Hydrochlorothiazide, HCTZ; Olmesartan
- Hydrochlorothiazide, HCTZ; Quinapril
- Hydrochlorothiazide, HCTZ; Spironolactone
- Hydrochlorothiazide, HCTZ; Telmisartan
- Hydrochlorothiazide, HCTZ; Triamterene
- Hydrochlorothiazide, HCTZ; Valsartan
- Hydrocodone; Ibuprofen
- Hydrocodone; Potassium Guaiacolsulfonate; Pseudoephedrine
- Hydrocodone; Pseudoephedrine
- Hydrocortisone
- Hyoscyamine
- Hyoscyamine; Methenamine; Methylene Blue; Phenyl Salicylate; Sodium Biphosphate
- Ibuprofen
- Ibuprofen; Oxycodone
- Ibuprofen; Pseudoephedrine
- Indacaterol; Glycopyrrolate
- Indomethacin
- Interferon Alfa-2a
- Interferon Alfa-2b
- Interferon Alfa-2b; Ribavirin
- Interferon Alfa-n3
- Interferon Alfacon-1
- Irbesartan
- Iron
- Ketoprofen
- Ketorolac
- Lansoprazole; Naproxen
- Lepirudin
- Lisinopril
- Lithium
- Loperamide
- Loperamide; Simethicone
- Loratadine; Pseudoephedrine
- Losartan
- Magnesium
- Magnesium Hydroxide
- Magnesium Salicylate
- Magnesium Salts
- Meclofenamate Sodium
- Mefenamic Acid
- Meloxicam
- Memantine
- Mepenzolate
- Methadone
- Methenamine
- Methenamine; Sodium Acid Phosphate
- Methenamine; Sodium Acid Phosphate; Methylene Blue; Hyoscyamine
- Methscopolamine
- Methyldopa
- Methylprednisolone
- Moexipril
- Mometasone
- Nabumetone
- Naproxen
- Naproxen; Pseudoephedrine
- Naproxen; Sumatriptan
- Nebivolol; Valsartan
- Nonsteroidal antiinflammatory drugs
- Olmesartan
- Oxaprozin
- Oxybutynin
- Palifermin
- Pegfilgrastim
- Peginterferon Alfa-2a
- Peginterferon Alfa-2b
- Penicillamine
- Penicillin G
- Pentosan
- Perindopril
- Perindopril; Amlodipine
- Piroxicam
- Platelet Inhibitors
- Potassium-sparing diuretics
- Prasugrel
- Prednisolone
- Prednisone
- Propantheline
- Pseudoephedrine
- Quinapril
- Quinidine
- Quinine
- Ramipril
- Reteplase, r-PA
- Rivaroxaban
- Rofecoxib
- Sacubitril; Valsartan
- Salsalate
- Scopolamine
- Sevelamer
- Sodium Polystyrene Sulfonate
- Spironolactone
- Streptokinase
- Sucralfate
- Sulfamethoxazole; Trimethoprim, SMX-TMP, Cotrimoxazole
- Sulindac
- Tacrolimus
- Tbo-Filgrastim
- Telmisartan
- Tenecteplase
- Thrombolytic Agents
- Ticagrelor
- Ticlopidine
- Tinzaparin
- Tirofiban
- Tolmetin
- Tolvaptan
- Trandolapril
- Trandolapril; Verapamil
- Triamcinolone
- Triamterene
- Trientine
- Trihexyphenidyl
- Trimethoprim
- Tuberculin Purified Protein Derivative, PPD
- Urokinase
- Valdecoxib
- Valsartan
- Vitamin D
- Vitamin D analogs
- Vorapaxar
- Warfarin
- Zinc
- Zinc Salts