Ioversol

Ioversol Brand Names

Optiray | Optiray-300 | Optiray-320 | Optiray-350

What is Ioversol

Loversol is an iodinated nonionic, low-osmolar contrast medium used for visualization of the internal structures of the body during angiography including digital subtraction angiography and excretory urography.

Ioversol is used to enhance computed tomography imaging of the head and body.

Ioversol was approved by the FDA on December 30, 1988.

Indications

  • angiography
  • computed tomography (CT) imaging
  • digital subtraction angiography (DSA)
  • urography

Side Effects

  1. abdominal pain
  2. acute generalized exanthematous pustulosis (AGEP)
  3. anaphylactic shock
  4. anaphylactoid reactions
  5. angina
  6. angioedema
  7. anuria
  8. anxiety
  9. aphasia
  10. apnea
  11. arachnoiditis
  12. asthenia
  13. AV block
  14. back pain
  15. bleeding
  16. blurred vision
  17. bradycardia
  18. bronchospasm
  19. cardiac arrest
  20. chest pain (unspecified)
  21. chills
  22. coma
  23. confusion
  24. conjunctivitis
  25. cough
  26. cyanosis
  27. disseminated intravascular coagulation (DIC)
  28. dizziness
  29. Drug Reaction with Eosinophilia and Systemic Symptoms (DRESS)
  30. dysgeusia
  31. dysphagia
  32. dyspnea
  33. ecchymosis
  34. erythema
  35. erythema multiforme
  36. fatigue
  37. fever
  38. flushing
  39. hallucinations
  40. headache
  41. hematoma
  42. hot flashes
  43. hyperhidrosis
  44. hypertension
  45. hypertensive crisis
  46. hyperthermia
  47. hyperthyroidism
  48. hyperventilation
  49. hypotension
  50. hypothyroidism
  51. hypoxia
  52. injection site reaction
  53. laryngeal edema
  54. laryngospasm
  55. maculopapular rash
  56. malaise
  57. metabolic acidosis
  58. myocardial infarction
  59. nasal congestion
  60. nausea
  61. oliguria
  62. palpitations
  63. paresis
  64. paresthesias
  65. peripheral edema
  66. peripheral vasodilation
  67. petechiae
  68. phlebitis
  69. polyuria
  70. pruritus
  71. pulmonary edema
  72. rash
  73. renal failure (unspecified)
  74. renal tubular necrosis
  75. respiratory arrest
  76. retroperitoneal bleeding
  77. rhabdomyolysis
  78. rhinitis
  79. seizures
  80. sinus tachycardia
  81. skin necrosis
  82. sneezing
  83. Stevens-Johnson syndrome
  84. stroke
  85. syncope
  86. thromboembolism
  87. thrombosis
  88. thyrotoxicosis
  89. tinnitus
  90. tissue necrosis
  91. toxic epidermal necrolysis
  92. tremor
  93. urinary retention
  94. urticaria
  95. ventricular fibrillation
  96. vertigo
  97. visual impairment
  98. vomiting
  99. weakness
  100. wheezing
  101. xerostomia

Monitoring Parameters

  • serum creatinine/BUN

Contraindications

  • asthma
  • atopy
  • breast-feeding
  • cardiac disease
  • children
  • coagulopathy
  • dehydration
  • diabetes mellitus
  • emphysema
  • extravasation
  • females
  • geriatric
  • heart failure
  • hepatic disease
  • hyperthyroidism
  • hypothyroidism
  • infants
  • intrathecal administration
  • iodine hypersensitivity
  • multiple myeloma
  • myasthenia gravis
  • neonates
  • pheochromocytoma
  • pregnancy
  • premature neonates
  • pulmonary disease
  • pulmonary hypertension
  • QT prolongation
  • radiopaque contrast media hypersensitivity
  • renal disease
  • renal failure
  • renal impairment
  • serious rash
  • sickle cell disease
  • thromboembolic disease
  • thyroid disease
  • thyrotoxicosis
  • valvular heart disease

Interactions

  • Acebutolol
  • Acetaminophen; Aspirin, ASA; Caffeine
  • Acetaminophen; Butalbital; Caffeine
  • Acetaminophen; Butalbital; Caffeine; Codeine
  • Acetaminophen; Caffeine
  • Acetaminophen; Caffeine; Dihydrocodeine
  • Acetaminophen; Caffeine; Magnesium Salicylate; Phenyltoloxamine
  • Acetaminophen; Caffeine; Phenyltoloxamine; Salicylamide
  • Acetaminophen; Chlorpheniramine; Dextromethorphan; Phenylephrine
  • Acetaminophen; Chlorpheniramine; Phenylephrine; Phenyltoloxamine
  • Acetaminophen; Dextromethorphan; Guaifenesin; Phenylephrine
  • Acetaminophen; Dextromethorphan; Phenylephrine
  • Acetaminophen; Guaifenesin; Phenylephrine
  • Acetaminophen; Tramadol
  • Acyclovir
  • Aldesleukin, IL-2
  • Alogliptin; Metformin
  • Aminoglycosides
  • Amiodarone
  • Amitriptyline
  • Amitriptyline; Chlordiazepoxide
  • Amoxapine
  • Amphetamine
  • Amphetamine; Dextroamphetamine
  • Amphetamine; Dextroamphetamine Salts
  • Amphotericin B
  • Angiotensin-converting enzyme inhibitors
  • Aprotinin
  • Aripiprazole
  • Asenapine
  • Aspirin, ASA; Butalbital; Caffeine
  • Aspirin, ASA; Butalbital; Caffeine; Codeine
  • Aspirin, ASA; Caffeine; Dihydrocodeine
  • Aspirin, ASA; Caffeine; Orphenadrine
  • Atenolol
  • Atenolol; Chlorthalidone
  • Bendroflumethiazide; Nadolol
  • Benzphetamine
  • Beta-blockers
  • Betaxolol
  • Bictegravir; Emtricitabine; Tenofovir Alafenamide
  • Bisoprolol
  • Bisoprolol; Hydrochlorothiazide, HCTZ
  • Brexpiprazole
  • Brimonidine; Timolol
  • Brompheniramine; Carbetapentane; Phenylephrine
  • Brompheniramine; Dextromethorphan; Phenylephrine
  • Bumetanide
  • Bupropion
  • Bupropion; Naltrexone
  • Caffeine
  • Caffeine; Ergotamine
  • Canagliflozin; Metformin
  • Capreomycin
  • Carbetapentane; Chlorpheniramine; Phenylephrine
  • Carbetapentane; Diphenhydramine; Phenylephrine
  • Carbetapentane; Guaifenesin; Phenylephrine
  • Carbetapentane; Phenylephrine
  • Carbetapentane; Phenylephrine; Pyrilamine
  • Carbinoxamine; Hydrocodone; Phenylephrine
  • Carbinoxamine; Phenylephrine
  • Carteolol
  • Carvedilol
  • Chlophedianol; Guaifenesin; Phenylephrine
  • Chlorpheniramine; Dextromethorphan; Phenylephrine
  • Chlorpheniramine; Dihydrocodeine; Phenylephrine
  • Chlorpheniramine; Hydrocodone; Phenylephrine
  • Chlorpheniramine; Phenylephrine
  • Cisplatin
  • Clomipramine
  • Clozapine
  • Cocaine
  • Codeine; Phenylephrine; Promethazine
  • Colistimethate, Colistin, Polymyxin E
  • Cyclobenzaprine
  • Cyclosporine
  • Dapagliflozin; Metformin
  • Darunavir; Cobicistat; Emtricitabine; Tenofovir alafenamide
  • Deferasirox
  • Desipramine
  • Dexmethylphenidate
  • Dextroamphetamine
  • Dextromethorphan; Diphenhydramine; Phenylephrine
  • Dextromethorphan; Guaifenesin; Phenylephrine
  • Diethylpropion
  • Diphenhydramine; Hydrocodone; Phenylephrine
  • Diphenhydramine; Phenylephrine
  • Dopamine
  • Doravirine; Lamivudine; Tenofovir disoproxil fumarate
  • Dorzolamide; Timolol
  • Doxepin
  • Efavirenz; Emtricitabine; Tenofovir
  • Efavirenz; Lamivudine; Tenofovir Disoproxil Fumarate
  • Elvitegravir; Cobicistat; Emtricitabine; Tenofovir Alafenamide
  • Elvitegravir; Cobicistat; Emtricitabine; Tenofovir Disoproxil Fumarate
  • Empagliflozin; Linagliptin; Metformin
  • Empagliflozin; Metformin
  • Emtricitabine; Rilpivirine; Tenofovir alafenamide
  • Emtricitabine; Rilpivirine; Tenofovir disoproxil fumarate
  • Emtricitabine; Tenofovir alafenamide
  • Emtricitabine; Tenofovir disoproxil fumarate
  • Entecavir
  • Ephedrine
  • Ertugliflozin; Metformin
  • Esmolol
  • Ethacrynic Acid
  • Ethanol
  • Fluoxetine; Olanzapine
  • Furosemide
  • Glipizide; Metformin
  • Glyburide; Metformin
  • Green Tea
  • Guaifenesin; Phenylephrine
  • Haloperidol
  • Hydrochlorothiazide, HCTZ; Metoprolol
  • Hydrochlorothiazide, HCTZ; Propranolol
  • Hydrocodone; Phenylephrine
  • Ibandronate
  • Iloperidone
  • Imipramine
  • Labetalol
  • Lamivudine; Tenofovir Disoproxil Fumarate
  • Levobetaxolol
  • Levobunolol
  • Linagliptin; Metformin
  • Lisdexamfetamine
  • Loop diuretics
  • Loxapine
  • Lurasidone
  • Maprotiline
  • Metformin
  • Metformin; Pioglitazone
  • Metformin; Repaglinide
  • Metformin; Rosiglitazone
  • Metformin; Saxagliptin
  • Metformin; Sitagliptin
  • Methamphetamine
  • Methylphenidate
  • Metoprolol
  • Midodrine
  • Molindone
  • Monoamine oxidase inhibitors
  • Nadolol
  • Nebivolol
  • Nebivolol; Valsartan
  • Nonsteroidal antiinflammatory drugs
  • Norepinephrine
  • Nortriptyline
  • Olanzapine
  • Oxaliplatin
  • Pamidronate
  • Pemoline
  • Penbutolol
  • Perphenazine; Amitriptyline
  • Phendimetrazine
  • Phenothiazines
  • Phentermine
  • Phentermine; Topiramate
  • Phenylephrine
  • Phenylephrine; Promethazine
  • Pimozide
  • Pindolol
  • Polymyxins
  • Propranolol
  • Protriptyline
  • Quetiapine
  • Risperidone
  • Sodium Iodide
  • Sodium Oxybate
  • Sotalol
  • Telbivudine
  • Tenofovir Alafenamide
  • Tenofovir Alafenamide
  • Tenofovir, PMPA
  • Thiothixene
  • Thyroid hormones
  • Timolol
  • Torsemide
  • Tramadol
  • Tricyclic antidepressants
  • Trimipramine
  • Valacyclovir
  • Ziprasidone
  • Zoledronic Acid
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